| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MC3R |
(R)-4-Amino-4-(naphthalen-2-ylmethyl-naphthalen-1-ylmethyl-carbamoyl)-butyric acid |
294000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
4-Naphthalen-2-ylmethyl-piperazine-1-carboxamidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N*1*-(1H-Indol-3-ylmethyl)-propane-1,3-diamine |
145000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
naphth-2-ylmethyl-Arg-Trp-NH2 |
107000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(S)-5-Guanidino-2-[(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amino]-pentanoic acid amide |
155000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
naphth-2-ylmethyl-D-Arg-Trp-NH2 |
147000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(2S)-N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-(1H-indol-3-ylmethylamino)pentanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(R)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid amide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2-yl-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(2S,4S)-4-hydroxy-N-[2-(1H-imidazol-5-yl)ethyl]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide |
161000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(R)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2-yl-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
prop-2-enyl (2S)-5-amino-2-(naphthalen-2-ylmethylamino)pentanoate |
161000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-[(2R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-oxidopiperazin-4-ium-1-yl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide |
114000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(4-(diethylamino)benzyl)-4-(1H-indol-3-yl)-N-pentylbutanamide |
289000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(3-aminopropyl)-N-(1-(benzo[b]thiophen-3-yl)ethyl)-4-(1H-indol-3-yl)butanamide |
104000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(3-aminopropyl)-N-cinnamyl-1H-indole-3-carboxamide |
172000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(3-aminopropyl)-5-(benzyloxy)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-indole-2-carboxamide |
542000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(4-aminobutyl)-N-isopropyl-1H-indole-3-carboxamide |
112000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
2-(4-hydroxybenzyl)-N-(4-aminobutyl)-N-isopropyl-1H-indole-3-carboxamide |
106000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(R)-2-amino-N-(5-aminopentyl)-N-benzyl-3-(4-nitrophenyl)propanamide |
162000 |
NA |
NA |
NA |
NA |
NA |
TTD |