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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MC3R (R)-2-amino-N-(5-aminopentyl)-N-benzyl-3-(1H-indol-3-yl)propanamide 106000 NA NA NA NA NA TTD
MC3R N-(4-(methylthio)benzyl)-N-(4-((4-aminocyclohexyl)methyl)cyclohexyl)-4-(1H-indol-3-yl)butanamide 249000 NA NA NA NA NA TTD
MC3R N-(4-(methylthio)benzyl)-4-(2-(4-hydroxybenzyl)-1H-indol-3-yl)-N-(4-((4-aminocyclohexyl)methyl)cyclohexyl)butanamide 201000 NA NA NA NA NA TTD
MC3R N-{4-[(4-aminocyclohexyl)methyl]cyclohexyl}-4-(1H-indol-3-yl)-N-[(2-methylphenyl)methyl]butanamide 121000 NA NA NA NA NA TTD
MC3R N-{4-[(4-aminocyclohexyl)methyl]cyclohexyl}-4-{2-[(4-hydroxyphenyl)methyl]-1H-indol-3-yl}-N-[(2-methylphenyl)methyl]butanamide 349000 NA NA NA NA NA TTD
MC3R N-{4-[(4-aminocyclohexyl)methyl]cyclohexyl}-4-(1H-indol-3-yl)-N-[(4-methylphenyl)methyl]butanamide 220000 NA NA NA NA NA TTD
MC3R N-{4-[(4-aminocyclohexyl)methyl]cyclohexyl}-4-{2-[(4-hydroxyphenyl)methyl]-1H-indol-3-yl}-N-[(4-methylphenyl)methyl]butanamide 147000 NA NA NA NA NA TTD
MC3R N-(3-bromo-4-methoxybenzyl)-4-(2-(4-hydroxybenzyl)-1H-indol-3-yl)-N-(4-((4-aminocyclohexyl)methyl)cyclohexyl)butanamide 132000 NA NA NA NA NA TTD
MC3R N-(4-((4-aminocyclohexyl)methyl)cyclohexyl)-4-(1H-indol-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)butanamide 278000 NA NA NA NA NA TTD
MC3R N-(2-guanidino-ethyl)-4-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-butyramide 204000 NA NA NA NA NA TTD
MC3R N-(3-guanidino-propyl)-2-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-acetamide 228000 NA NA NA NA NA TTD
MC3R N-(4-guanidino-butyl)-2-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-acetamide 137000 NA NA NA NA NA TTD
MC3R N-(4-guanidino-butyl)-4-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-butyramide 134000 NA NA NA NA NA TTD
MC3R Cefepime NA NA NA NA NA 300000 PubChem
MC3R Ceftazidime NA NA NA NA NA 300000 PubChem
MC3R Aztreonam NA NA NA NA NA 400000 PubChem
MC3R Carumonam NA NA NA NA NA 500000 PubChem
MC3R (2R)-N-(1H-indol-3-ylmethyl)-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide 104000 NA NA NA NA NA TTD
MC3R (2R)-1-[2-(1H-indol-3-yl)ethyl]-N-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide 752000 NA NA NA NA NA TTD
MC3R Doripenem NA NA NA NA NA 300000 PubChem