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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MC4R prop-2-enyl (2S)-5-amino-2-(naphthalen-2-ylmethylamino)pentanoate 127000 NA NA NA NA NA TTD
MC4R (S)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-amino]-propionamide 139000 NA NA NA NA NA TTD
MC4R N-[(2R)-3-(4-chlorophenyl)-1-(4-oxido-4-phenylpiperazin-4-ium-1-yl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 169000 NA NA NA NA NA TTD
MC4R N-(2-aminoethyl)-N-cinnamyl-3-(1H-indol-3-yl)propanamide 106000 NA NA NA NA NA TTD
MC4R N-(3-aminopropyl)-4-(1H-indol-3-yl)-N-phenethylbutanamide 164000 NA NA NA NA NA TTD
MC4R N-(4-aminobutyl)-3-(1H-indol-3-yl)-N-(1-phenylpropyl)propanamide 158000 NA NA NA NA NA TTD
MC4R N-(4-aminobutyl)-N-isopropyl-1H-indole-3-carboxamide 222000 NA NA NA NA NA TTD
MC4R 2-(4-hydroxybenzyl)-N-(4-aminobutyl)-N-isopropyl-1H-indole-3-carboxamide 165000 NA NA NA NA NA TTD
MC4R N-(2-guanidino-ethyl)-2-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-acetamide 179000 NA NA NA NA NA TTD
MC4R N-(2-carbamimidamidoethyl)-3-(1H-indol-3-yl)-N-(naphthalen-2-ylmethyl)propanamide 149000 NA NA NA NA NA TTD
MC4R N-(2-guanidino-ethyl)-4-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-butyramide 179000 NA NA NA NA NA TTD
MC4R N-(3-guanidino-propyl)-2-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-acetamide 150000 NA NA NA NA NA TTD
MC4R N-(4-guanidino-butyl)-2-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-acetamide 182000 NA NA NA NA NA TTD
MC4R N-(4-guanidino-butyl)-3-(1H-indol-3-yl)-N-naphthalen-2-ylmethyl-propionamide 116000 NA NA NA NA NA TTD
MC4R N-((1R,2R)-2-aminocyclohexyl)-N-cinnamyl-4-(1H-indol-3-yl)butanamide 116000 NA NA NA NA NA TTD
MC4R (2R)-1-[2-(1H-indol-3-yl)ethyl]-N-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide 166000 NA NA NA NA NA TTD
MC4R 1-(Naphthalen-2-ylmethyl)piperazine 1000000 NA NA NA NA NA TTD
MC4R N-(2-aminoethyl)-2-(1H-indol-3-yl)-N-(naphthalen-2-ylmethyl)acetamide 140000 NA NA NA NA NA TTD
MC5R N-(3-aminopropyl)-2-(naphthalen-2-yl)-N-(naphthalen-2-ylmethyl)acetamide 267000 NA NA NA NA NA TTD
MC5R 3-(piperazin-1-ylmethyl)-1H-indole 256000 NA NA NA NA NA TTD