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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MC3R 1-(Naphthalen-2-ylmethyl)piperazine 1000000 NA NA NA NA NA TTD
MC3R N-(2-aminoethyl)-3-(1H-indol-3-yl)-N-(3-phenylpropyl)propanamide 127000 NA NA NA NA NA TTD
MC4R N-(3-aminopropyl)-2-(1H-indol-3-yl)-N-(naphthalen-2-ylmethyl)acetamide 161000 NA NA NA NA NA TTD
MC4R N-(4-aminobutyl)-2-(1H-indol-3-yl)-N-(naphthalen-2-ylmethyl)acetamide 111000 NA NA NA NA NA TTD
MC4R 3-(piperazin-1-ylmethyl)-1H-indole 1000000 NA NA NA NA NA TTD
MC4R 2-(1H-indol-3-yl)-N-(1H-indol-3-ylmethyl)ethanamine 161000 NA NA NA NA NA TTD
MC4R N-(1-naphthylmethyl)-N-(2-naphthylmethyl)amine 1000000 NA NA NA NA NA TTD
MC4R 2-(1H-indol-3-yl)-N-(naphthalen-2-ylmethyl)ethanamine 118000 NA NA NA NA NA TTD
MC4R 4-(1H-Indol-3-ylmethyl)-piperazine-1-carboxamidine 1000000 NA NA NA NA NA TTD
MC4R (1H-Indol-3-ylmethyl)-naphthalen-1-ylmethyl-amine 161000 NA NA NA NA NA TTD
MC4R N-{3-[(1H-Indol-3-ylmethyl)-amino]-propyl}-guanidine 107000 NA NA NA NA NA TTD
MC4R N*1*-(1H-Indol-3-ylmethyl)-propane-1,3-diamine 104000 NA NA NA NA NA TTD
MC4R naphth-2-ylmethyl-Arg-Trp-NH2 105000 NA NA NA NA NA TTD
MC4R (S)-5-Guanidino-2-[(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amino]-pentanoic acid amide 134000 NA NA NA NA NA TTD
MC4R (2S)-N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-(1H-indol-3-ylmethylamino)pentanamide 205000 NA NA NA NA NA TTD
MC4R (R)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid amide 1000000 NA NA NA NA NA TTD
MC4R (2S,4S)-N-[3-(diaminomethylideneamino)propyl]-4-hydroxy-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide 279000 NA NA NA NA NA TTD
MC4R (S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2-yl-propionamide 1000000 NA NA NA NA NA TTD
MC4R (2S,4S)-4-hydroxy-N-[2-(1H-imidazol-5-yl)ethyl]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide 150000 NA NA NA NA NA TTD
MC4R (R)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2-yl-propionamide 1000000 NA NA NA NA NA TTD