| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MC1R |
N-(1-naphthylmethyl)-N-(2-naphthylmethyl)amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
4-(1H-Indol-3-ylmethyl)-piperazine-1-carboxamidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
N*1*-Naphthalen-2-ylmethyl-propane-1,3-diamine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
4-Naphthalen-2-ylmethyl-piperazine-1-carboxamidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
(S)-5-Guanidino-2-[(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amino]-pentanoic acid amide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
(2S)-N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-(1H-indol-3-ylmethylamino)pentanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
(R)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid amide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
N-[(2R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-oxidopiperazin-4-ium-1-yl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide |
152000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC1R |
(1R,4S,6R)-N-[(2R)-1-[4-(tert-butylcarbamoyl)-4-cyclohexylpiperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]-7-methyl-7-azabicyclo[2.2.2]octane-6-carboxamide |
NA |
NA |
NA |
160000 |
NA |
NA |
TTD |
| MC1R |
1-(Naphthalen-2-ylmethyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(2-aminoethyl)-N-(naphthalen-2-ylmethyl)-1H-indole-3-carboxamide |
134000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(3-aminopropyl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-indole-3-carboxamide |
131000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| MC3R |
3-(piperazin-1-ylmethyl)-1H-indole |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
N-(1-naphthylmethyl)-N-(2-naphthylmethyl)amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| MC3R |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| MC3R |
4-(1H-Indol-3-ylmethyl)-piperazine-1-carboxamidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(1H-Indol-3-ylmethyl)-naphthalen-1-ylmethyl-amine |
214000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MC3R |
(2S)-N-(4-aminobutyl)-6-(1H-indol-3-ylmethylamino)-2-(naphthalen-2-ylmethylamino)hexanamide |
167000 |
NA |
NA |
NA |
NA |
NA |
TTD |