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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MCL1 2-Hydroxy-5-(methylsulfanyl)benzoic acid NA 160000 NA NA NA NA BindingDB|ChEMBL|TTD
MCL1 3,6,7-Trimethyl-benzofuran-2-carboxylic acid 214000 NA NA NA NA NA BindingDB|ChEMBL|TTD
MCL1 1,2-Acenaphthylenedione NA NA|1425000 324690|NA|323593.66 NA NA NA BindingDB|ChEMBL
MCL1 1-(3-Naphthalen-1-yloxypropyl)indole-2-carboxamide 500000 NA NA NA NA NA TTD
MCL1 5-naphthalen-1-yl-2-oxo-1H-pyridine-3-carbonitrile NA 158500 NA NA NA NA BindingDB|ChEMBL
MCL1 2-oxo-5-(4-phenylphenyl)-1H-pyridine-3-carbonitrile NA 316200 NA NA NA NA BindingDB|ChEMBL
MCL1 5-[4-(2-methylbutan-2-yl)phenyl]sulfanyl-2-oxo-1H-pyridine-3-carbonitrile NA 177500 NA NA NA NA BindingDB|ChEMBL
MCL1 5-(4-bromophenyl)sulfanyl-2-oxo-1H-pyridine-3-carbonitrile NA 121100 NA NA NA NA BindingDB|ChEMBL
MCL1 5-(4-aminophenyl)sulfanyl-2-oxo-1H-pyridine-3-carbonitrile NA 133300 NA NA NA NA BindingDB|ChEMBL
MCL1 1-Benzyl-2-oxo-5-(4-propan-2-ylphenyl)sulfanylpyridine-3-carbonitrile NA 383100 NA NA NA NA BindingDB
MCL1 Indole-2-carboxylic acid 1000000 NA NA NA NA NA TTD
MCL1 Cyanoacetamide NA NA 1000000 NA NA NA PubChem
MCL1 2-[5-[(4-Bromophenyl)sulfonylamino]-2-hydroxyphenyl]sulfanylacetic acid 283360 NA NA NA NA NA BindingDB
MCL1 Ethyl 2-Amino-6-(3'',5''-dimethoxyphenyl)-4-(2-ethoxy-2-oxoethyl)-4H-chromene-3-carboxylate 41999000 NA NA NA NA NA BindingDB
MCL1 3-[5-[(1,3-Benzothiazol-2-yldiazenyl)methyl]furan-2-yl]-2-methylbenzoic acid NA 167000 NA NA NA NA BindingDB
MCL1 2-(4-Chloro-3-methylphenoxy)acetic acid 103000 NA NA NA NA NA BindingDB|ChEMBL|TTD
MDH1 Benzyl Benzoate NA 125000 NA NA NA NA BindingDB|PubChem
MDH1 Fluconazole NA 400000 NA NA NA NA PubChem
MDH1 Glyburide NA 400000 NA NA NA NA BindingDB|PubChem
MDH1 1-[4-[4-[[2-(2,4-Dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]ethanone NA 150000 NA NA NA NA PubChem