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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MMP8 (2S)-2-[(4-nitrophenyl)sulfonylamino]-5-oxo-5-(pentylamino)pentanoic acid NA 500000 NA NA NA NA TTD
MMP8 (2S)-5-(methylamino)-2-[(4-nitrophenyl)sulfonylamino]-5-oxopentanoic acid NA 401100 NA NA NA NA BindingDB|TTD
MMP8 (2S)-5-(2-methylpropylamino)-2-[(4-nitrophenyl)sulfonylamino]-5-oxopentanoic acid NA 483100 NA NA NA NA BindingDB|TTD
MMP8 (2S)-2-[(4-nitrophenyl)sulfonylamino]-5-oxo-5-(propan-2-ylamino)pentanoic acid NA 500000 NA NA NA NA TTD
MMP8 (2S)-5-amino-2-[(4-nitrophenyl)sulfonylamino]-5-oxopentanoic acid NA 198900 NA NA NA NA BindingDB|TTD
MMP8 (2S)-5-(butylamino)-2-[(4-nitrophenyl)sulfonylamino]-5-oxopentanoic acid NA 345800 NA NA NA NA BindingDB|TTD
MMP8 (2S)-5-(benzylamino)-2-[(4-nitrophenyl)sulfonylamino]-5-oxopentanoic acid NA 172800 NA NA NA NA BindingDB|TTD
MMP8 (2S)-5-(ethylamino)-2-[(4-nitrophenyl)sulfonylamino]-5-oxopentanoic acid NA 298500 NA NA NA NA BindingDB|TTD
MMP8 D-Leucyl-L-phenylalanine methylamide NA 300000 NA NA NA NA TTD
MMP8 2-[5-(4-Fluorophenyl)-2-[4-[4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]-3,4-dihydropyrazol-3-yl]phenol NA 100100 NA NA NA NA BindingDB|TTD
MMP8 4-[[2-(4-Bromophenyl)acetyl]amino]-5-[(4-nitrophenyl)methylamino]-5-oxopentanoic acid NA 205890 NA NA NA NA BindingDB
MMP8 N-[(Hydroxyamino)carbonyl]-D-leucyl-Lphenylalanine methylamide NA 150000 NA NA NA NA BindingDB|TTD
MMP8 Nafamostat NA 420000 NA NA NA NA PubChem
MMP8 1-[2-[4-(4-Cyanophenyl)phenoxy]ethyl]-3-hydroxyurea NA 120000 NA NA NA NA TTD
MMP8 (1-Benzyloxycarbonylamino-2-phenyl-ethyl)-[2-[1-carbamoyl-2-(1H-indol-3-yl)-ethylcarbamoyl]-3-(2-trifluoromethoxy-phenylsulfanyl)-propyl]-phosphinic acid 200000 NA NA NA NA NA BindingDB|TTD
MMP8 1-(2-Hydroxycarbamoyl-4-methyl-pentanoyl)-pyrrolidine-2-carboxylic acid benzylamide 168000 NA NA NA NA NA BindingDB|TTD
MMP8 N-Benzyl-3-(2-hydroxycarbamoyl-4-methyl-pentanoylamino)-succinamic acid 136000 NA NA NA NA NA BindingDB
MMP8 1-(4-Phenoxyphenethyl)-3-hydroxyurea NA 380000 NA NA NA NA TTD
MMP8 1-(4-Phenoxyphenethyl)-3-hydroxy-1-methylurea NA 1000000 NA NA NA NA BindingDB|TTD
MMP8 Ethyl 2-(hydroxycarbamoyl)-3-methylbutanoate 190546|190546.07 NA NA NA NA NA BindingDB|TTD