| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MMP3 |
N-[(1S,2S)-2-sulfanylcyclopentyl]benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
4-phenoxy-N-[(1S,2S)-2-sulfanylcyclopentyl]benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-[(1S,2S)-2-hydroxycyclopentyl]-4-phenoxybenzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
4-phenoxy-N-[(1S,2S)-2-sulfanylcyclopentyl]benzamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(R)-2-(((benzyloxy)carbonyl)amino)-3-(4-hydroxyphenyl)propanoic acid |
356000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-Acetyl-D-tyrosine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
benzyl N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]carbamate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
D-Tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Fmoc-L-tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Fmoc-D-Trp-OH |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1,3,2,6-Tetraguanidinoneamine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP7 |
(1S,2R)-2-cyano-N-hydroxy-2-(4-((2-phenylquinolin-4-yl)methoxy)benzyl)cyclopropanecarboxamide |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP7 |
N-(4-(4-(thiiran-2-ylmethylsulfonyl)phenoxy)phenyl)methanesulfonamide |
295000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MMP7 |
(1S,5S,7R)-N~7~-(Biphenyl-4-ylmethyl)-N~3~-hydroxy-6,8-dioxa-3-azabicyclo(3.2.1)octane-3,7-dicarboxamide |
NA |
1510000 |
NA |
NA |
NA |
NA |
BindingDB |
| MMP7 |
N-benzyloxycarbonyl-L-leucyl-L-phenylalanine methyl ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP7 |
D-Leucyl-L-phenylalanine methylamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP7 |
MMP-2 Inhibitor II |
379000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| MMP7 |
(2~{R})-2-[[4-[(4-aminocarbonylphenyl)carbonylamino]phenyl]sulfonylamino]-5-[(2~{S},4~{S})-4-azanyl-2-[[(2~{S})-1-[[(2~{S})-1-[(5-azanyl-5-oxidanylidene-pentyl)amino]-5-oxidanyl-1,5-bis(oxidanylidene)pentan-2-yl]-methyl-amino]-4-methyl-1-oxidanylidene-pentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxidanylidene-pentanoic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| MMP7 |
L-Leucyl-L-phenylalanine methylamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP7 |
(1S,2R)-1-N-hydroxy-2-({4-[(2-methylquinolin-4-yl)methoxy]phenyl}methyl)cyclopropane-1,2-dicarboxamide |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |