| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MMP3 |
(1S,2R)-N-hydroxy-2-((S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl)-2-(4-((2-phenylquinolin-4-yl)methoxy)benzyl)cyclopropanecarboxamide |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(1R,2S)-ethyl 2-(hydroxycarbamoyl)-1-(4-((2-methylquinolin-4-yl)methoxy)benzyl)cyclopropanecarboxylate |
952000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(1R,2S)-ethyl 2-(hydroxycarbamoyl)-1-(4-((2-phenylquinolin-4-yl)methoxy)benzyl)cyclopropanecarboxylate |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
5-(Ethylamino)-1,3,4-thiadiazole-2-thiol |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
5-[(2-Furylmethyl)amino]-1,3,4-thiadiazole-2-thiol |
NA |
289000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Salicylamide |
NA |
NA |
25000000 |
NA |
NA |
NA |
PubChem |
| MMP3 |
N-(2-((4'-Cyano-1,1'-biphenyl-4-YL)oxy)ethyl)-N'-hydroxy-N-methylurea |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Tetracycline |
NA |
140000 |
NA |
NA |
NA |
NA |
PubChem |
| MMP3 |
Minocycline |
NA |
290000 |
NA |
NA |
NA |
NA |
PubChem |
| MMP3 |
Tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| MMP3 |
N-(Benzyloxycarbonyl)-D-phenylalanine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-Acetyl-L-tyrosine |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| MMP3 |
(2Z,NE)-N-benzylidene-4-(3,4-dimethoxyphenyl)-2-(phenylimino)thiazol-3(2H)-amine |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Z-Tyr-NH2 |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-Acetyl-L-tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(S)-Benzyl (1-hydrazinyl-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)carbamate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-Benzoyl-L-Tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1,3,4-Thiadiazole-2(3H)-thione, 5-anilino- |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
4-Hydroxybiphenyl |
NA |
NA |
280000 |
NA |
NA |
NA |
ChEMBL |
| MMP3 |
4-phenoxy-N-[(1R,2S)-2-sulfanylcyclopentyl]benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |