| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MMP3 |
1-Ethyl-3-phenethyl-1-(5-thioxo-4,5-dihydro-[1,3,4]thiadiazol-2-yl)-urea |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-Methyl-2-[3-(5-thioxo-4,5-dihydro-[1,3,4]thiadiazol-2-yl)-ureido]-acetamide |
165958.69 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1-(4-Methyl-5-thioxo-4,5-dihydro-[1,3,4]thiadiazol-2-yl)-3-phenethyl-urea |
NA |
694000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1-Benzyl-3-[1,3,4]thiadiazol-2-yl-urea |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
5-(4-Phenyl-butylamino)-3H-[1,3,4]thiadiazole-2-thione |
NA |
318000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-((tert-Butoxy)carbonyl)-D-tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1,3,2-Triguanidinoneamine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(1S,2R)-2-cyano-N-hydroxy-2-(4-((2-phenylquinolin-4-yl)methoxy)benzyl)cyclopropanecarboxamide |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
L-Tyrosine, N-(1,1-dimethylethoxy)carbonyl- |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Berkchaetoazaphilone A |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(3E,5R,6S,15S,16R)-5,6,15-trihydroxy-16-methyl-1-oxacyclohexadec-3-en-2-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
4-[(5Z)-2,4-Dioxo-5-[(2E)-3-phenylprop-2-EN-1-ylidene]-1,3-thiazolidin-3-YL]butanoic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-benzyloxycarbonyl-L-leucyl-L-phenylalanine methyl ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
D-Leucyl-L-phenylalanine methylamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(2R)-2-(((tert-butoxy)carbonyl)amino)-3-(4-hydroxyphenyl)propanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Acetohydroxamic Acid |
NA |
NA |
17000000 |
NA |
NA |
NA |
PubChem |
| MMP3 |
(E)-2-(5-((5-(4-methoxyphenyl)furan-2-yl)methylene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid |
NA |
850000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-[1-(4''-Cyano-biphenyl-4-yloxymethyl)-2-(4-fluoro-phenyl)-ethyl]-N-hydroxy-formamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-[1-(4''-Cyano-biphenyl-4-yloxymethyl)-3-methyl-butyl]-N-hydroxy-formamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-[2-(4''-Cyano-biphenyl-4-yloxy)-1-(4-fluoro-phenyl)-ethyl]-N-hydroxy-formamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |