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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
MMP2 (2S)-N-hydroxy-4-methylsulfanyl-2-(2-phenylethylcarbamoylamino)butanamide NA 500000 NA NA NA NA TTD
MMP2 (2S)-2-[(4-fluorophenyl)methylcarbamoylamino]-N-hydroxy-4-methylpentanamide NA 1000000 NA NA NA NA TTD
MMP2 [(2S)-3-[[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-oxo-2-[2-(trifluoromethoxy)phenyl]sulfanylpropyl]-[(1R)-2-phenyl-1-(phenylmethoxycarbonylamino)ethyl]phosphinic acid 200000 NA NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-2-[(3-methoxyphenyl)methylcarbamoylamino]-4-methylpentanamide NA 1000000 NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-2-[(4-methoxyphenyl)methylcarbamoylamino]-4-methylpentanamide NA 1000000 NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-4-methyl-2-[(4-methylphenyl)carbamoylamino]pentanamide NA 573000 NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-2-[(2-methoxyphenyl)methylcarbamoylamino]-4-methylpentanamide NA 1000000 NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-2-[(4-methoxyphenyl)carbamoylamino]-4-methylpentanamide NA 1000000 NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-4-methyl-2-[(4-methylphenyl)methylcarbamoylamino]pentanamide NA 1000000 NA NA NA NA TTD
MMP2 (2S)-2-[(3-fluorophenyl)methylcarbamoylamino]-N-hydroxy-4-methylpentanamide NA 1000000 NA NA NA NA TTD
MMP2 (2S)-N-hydroxy-4-methyl-2-(naphthalen-1-ylcarbamoylamino)pentanamide NA 1000000 NA NA NA NA TTD
MMP2 Ubenimex NA 162000|276000|163480|156980|120400|156000|253200 NA NA NA NA PubChem
MMP2 2-[[4-[(3,5-Dibromophenyl)methoxy]phenyl]sulfonylamino]acetic acid NA 125000 NA NA NA NA TTD
MMP2 (8S)-7-(4-methylphenyl)sulfonyl-1,4-dithia-7-azaspiro[4.4]nonane-8-carbohydrazide NA 428990 NA NA NA NA TTD
MMP2 H-Tic-Thr-NHOH.HCl NA 200630 NA NA NA NA TTD
MMP2 H-Tic-Ile-NHOH.HCl NA 671560 NA NA NA NA TTD
MMP2 8-Mercaptoquinoline NA 200000 NA NA NA NA TTD
MMP2 [(4S,5S)-2-(4-Bromo-phenyl)-5-vinyl-4,5-dihydro-oxazol-4-yl]-methanol 600000 NA NA NA NA NA TTD
MMP3 N-[2-(4''-Cyano-biphenyl-4-yloxy)-1-methyl-ethyl]-N-hydroxy-formamide NA 620000 NA NA NA NA TTD
MMP3 (2R)-N-hydroxy-4-methyl-2-{[methyl(phenyl)phosphoryl]amino}pentanamide NA 130500 NA NA NA NA TTD