| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MMP3 |
N-[2-(4''-Cyano-biphenyl-4-yloxy)-1-phenoxymethyl-ethyl]-N-hydroxy-formamide |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
3,2-Diguanidinoneamine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1,3,2,6-Tetraguanidino-5,6,3,4-tetramethoxylneamine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-[(Hydroxyamino)carbonyl]-D-leucyl-Lphenylalanine methylamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-[(Hydroxyamino)carbonyl]-L-leucyl-Lphenylalanine methylamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Clodronic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| MMP3 |
Salicylic Acid |
NA |
NA |
25000000 |
NA |
NA |
NA |
PubChem |
| MMP3 |
4-(4-Methoxy-phenyl)-thiophene-2-carboxylic acid (2-morpholin-4-yl-ethyl)-amide |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
Hydroxyurea |
NA |
NA |
25000000 |
NA |
NA |
NA |
PubChem |
| MMP3 |
(S)-2-((E)-3-Furan-2-yl-acryloylamino)-3-(1H-indol-3-yl)-propionic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
3-(4-(2-oxo-2H-chromen-3-yl)-2-thioxo-2,3-dihydro-1H-imidazol-1-yl)benzoic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
N-acetyl-D-tryptophan |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1-(4-Chloro-2-methyl-phenyl)-3-(5-thioxo-4,5-dihydro-[1,3,4]thiadiazol-2-yl)-urea |
119000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
5-(2-Chloro-6-methyl-phenylamino)-3H-[1,3,4]thiadiazole-2-thione |
NA |
173000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(R)-2-[(S)-3-(4-Isopropyl-phenoxy)-1-((S)-6-methylcarbamoyl-tetrahydro-pyridazine-1-carbonyl)-propylamino]-propionic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(R)-2-[(S)-3-(4-Cyclopentylmethyl-phenoxy)-1-((S)-6-methylcarbamoyl-tetrahydro-pyridazine-1-carbonyl)-propylamino]-propionic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
[(2S)-1-[[(2S)-1-(benzylamino)-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]oxy-[4-(1,3-dioxoisoindol-2-yl)butyl]phosphinic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1-(4-Phenoxyphenethyl)-3-hydroxyurea |
NA |
380000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
1-(4-Phenoxyphenethyl)-3-hydroxy-1-methylurea |
NA |
380000 |
NA |
NA |
NA |
NA |
TTD |
| MMP3 |
(1R,2S)-1-(3-fluoro-4-((2-phenylquinolin-4-yl)methoxy)benzyl)-N2-hydroxy-N1,N1-dimethylcyclopropane-1,2-dicarboxamide |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |