| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NFE2L2 |
Phenol |
NA |
NA |
NA |
NA |
1000000 |
NA |
PubChem |
| NFKB1 |
4,6-dichloro-N-(4-chlorophenyl)-1,3,5-triazin-2-amine |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| NFKB1 |
4,6-Dichloro-N-(4-nitrophenyl)-1,3,5-triazin-2-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| NFKB1 |
4-{[(3-tert-butyl-5,9-dimethyl-7-oxo-7H-furo[3,2-g]chromen-6-yl)acetyl]amino}butanoic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| NFKB1 |
3-(3-tert-butyl-5,9-dimethyl-7-oxo-7H-furo[3,2-g]chromen-6-yl)-N-(2-chlorobenzyl)propanamide |
NA |
NA |
NA |
4000000 |
NA |
NA |
TTD |
| NFKB1 |
2-(3-tert-butyl-5,9-dimethyl-7-oxo-7H-furo[3,2-g]chromen-6-yl)-N-(2-chlorobenzyl)acetamide |
NA |
NA |
NA |
5000000 |
NA |
NA |
TTD |
| NFKB1 |
2-[[2-(3-Tert-butyl-5-methyl-7-oxofuro[3,2-g]chromen-6-yl)acetyl]amino]-3-phenylpropanoic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| NFKB1 |
2,4-Dichloro-6-(3-nitroanilino)-1,3,5-triazine |
NA |
119000 |
NA |
NA |
NA |
NA |
TTD |
| NFKB1 |
3-Phenyl-2-[[2-(2,3,5,9-tetramethyl-7-oxofuro[3,2-g]chromen-6-yl)acetyl]amino]propanoic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| NFKB1 |
3-Phenyl-2-[3-(2,3,5,9-tetramethyl-7-oxofuro[3,2-g]chromen-6-yl)propanoylamino]propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| NFKB1 |
2-[[2-(4,11-Dimethyl-2-oxo-6,7,8,9-tetrahydro-[1]benzofuro[3,2-g]chromen-3-yl)acetyl]amino]-3-phenylpropanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| NFKB1 |
N-[(2-Chlorophenyl)methyl]-2-{3,5,9-trimethyl-7-oxo-7H-furo[3,2-G]chromen-6-YL}acetamide |
NA |
NA |
NA |
800000 |
NA |
NA |
TTD |
| NFKB1 |
Hymecromone |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| NFKB1 |
2-Phenylphenol |
NA |
NA |
NA |
NA |
251189 |
NA |
PubChem |
| NFKB1 |
4-[[[2-(3-Tert-butyl-5-methyl-7-oxofuro[3,2-g]chromen-6-yl)acetyl]amino]methyl]benzoic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| NFKB1 |
2-[4-[[2-(3-Tert-butyl-5-methyl-7-oxofuro[3,2-g]chromen-6-yl)acetyl]amino]phenyl]acetic acid |
NA |
NA |
NA |
530000 |
NA |
NA |
TTD |
| NFKB1 |
4-[[3-(3-Tert-butyl-5-methyl-7-oxofuro[3,2-g]chromen-6-yl)propanoylamino]methyl]benzoic acid |
NA |
NA |
NA |
670000 |
NA |
NA |
TTD |
| NFKB1 |
3-[[2-(2,3,5-Trimethyl-7-oxofuro[3,2-g]chromen-6-yl)acetyl]amino]benzoic acid |
NA |
NA |
NA |
700000 |
NA |
NA |
TTD |
| NFKB1 |
3-[3-(2,3,5-Trimethyl-7-oxofuro[3,2-g]chromen-6-yl)propanoylamino]benzoic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| NFKB1 |
3-[[2-(2,3,5,9-Tetramethyl-7-oxofuro[3,2-g]chromen-6-yl)acetyl]amino]benzoic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |