| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NISCH |
5-(3-chloro-4-fluorophenyl)-3-diethoxyphosphoryl-3a,6a-dihydro-3H-pyrrolo[3,4-c]pyrrole-4,6-dione |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| NLRP3 |
(5S,6R)-5-hydroxy-6-(hydroxymethyl)oxan-3-one |
NA |
2300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NLRP3 |
Nlrp3/aim2-IN-3 |
NA |
NA |
1630000 |
NA |
NA |
NA |
BindingDB |
| NMT1 |
(E)-methyl 4-(4-chlorophenylamino)-4-oxobut-2-enoate |
NA |
400000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[4-(1-methylpiperidin-4-yl)butyl]-~{N}-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[4-(1-methylpiperidin-4-yl)butyl]benzenesulfonamide |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[3-[[(1R,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]oxy]propyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide |
NA |
130000|27000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[3-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]propyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide |
NA |
640000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[3-[[(1R,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]oxy]propyl]-N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]benzenesulfonamide |
NA |
12000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[4-[(3R,5S)-3,5-dimethylpiperazin-1-yl]butyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide |
NA |
10000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-[[(3R)-4-methylmorpholin-3-yl]methoxy]propyl]benzenesulfonamide |
NA |
9600000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[4-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]butyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide |
NA |
3600000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[3-(4-methyl-1,4-diazepan-1-yl)propyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-[[(2S)-1-methylpyrrolidin-2-yl]methoxy]propyl]benzenesulfonamide |
NA |
2500000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
N-[6-(2-methylpropyl)quinolin-5-yl]-4-(4-piperazin-1-ylbutyl)benzenesulfonamide |
NA |
2000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[3-(4-methyl-1,4-diazepan-1-yl)propyl]-N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]benzenesulfonamide |
NA |
290000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[4-(4-methyl-1,4-diazepan-1-yl)butyl]-N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]benzenesulfonamide |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-[[(2S)-4-methylmorpholin-2-yl]methoxy]propyl]benzenesulfonamide |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
4-[4-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]butyl]-N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]benzenesulfonamide |
NA |
13000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NMT1 |
N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-[[(2R)-1-methylpyrrolidin-2-yl]methoxy]propyl]benzenesulfonamide |
NA |
730000 |
NA |
NA |
NA |
NA |
BindingDB |