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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
NMT1 4-(3-tert-Butylamino-propoxy)-3-methyl-benzofuran-2-carboxylic acid ethyl ester NA 200000 NA NA NA NA BindingDB
NMT1 Ethyl 3-methyl-4-[3-(1-piperidyl)propoxy]benzofuran-2-carboxylate NA 170000 NA NA NA NA BindingDB
NMT1 Ethyl 3-methyl-4-{3-[benzylamino]propoxy}benzo[d]furan-2-carboxylate NA 530000 NA NA NA NA BindingDB
NMT1 Ethyl 3-ethyl-4-{3-[(3-pyridylmethyl)amino]propoxy}benzo[d]furan-2-carboxylate NA 280000 NA NA NA NA BindingDB
NMT1 Ethyl 3-(methylethyl)-4-{3-[(3-pyridylmethyl)amino]propoxy}benzo[d]furan-2-carboxylate NA 260000 NA NA NA NA BindingDB
NMT1 [3-Methyl-4-[3-(3-pyridylmethylamino)propoxy]benzofuran-2-yl]-(2-pyridyl)methanone NA 340000 NA NA NA NA BindingDB
NMT1 [3-Methyl-4-[3-(3-pyridylmethylamino)propoxy]benzofuran-2-yl]-(4-methylthiazol-2-yl)methanone NA 130000 NA NA NA NA BindingDB
NMT1 2-Furyl-[3-methyl-4-[3-(3-pyridylmethylamino)propoxy]benzofuran-2-yl]methanone NA 150000|280000 NA NA NA NA BindingDB
NMT1 (2E)-4-[(4-nitrophenyl)amino]-4-oxobut-2-enoic acid NA 2560000 NA NA NA NA BindingDB
NMT1 4-Bromo-2-methyl-N-(1,3,5-trimethyl-1H-pyrazol-4-yl)-benzenesulfonamide NA 107000 NA NA NA NA BindingDB
NMT1 (2E)-4-[(3,4-Dimethylphenyl)amino]-4-oxobut-2-enoic acid NA 7550000 NA NA NA NA BindingDB
NMT1 4-(4-Chloroanilino)-4-oxobut-2-enoic acid NA 1600000 NA NA NA NA BindingDB
NMT1 (2E)-4-((4-Methylphenyl)amino)-4-oxo-2-butenoic acid NA 8350000 NA NA NA NA BindingDB
NMT1 (2E)-4-[(3,4-dichlorophenyl)amino]-4-oxobut-2-enoic acid NA 4380000 NA NA NA NA BindingDB
NMT1 (2S)-2-[[(2S)-6-amino-2-[[(2S)-3-hydroxy-2-[2-[4-[4-(2-methylimidazol-1-yl)butyl]phenyl]propanoylamino]propanoyl]amino]hexanoyl]amino]-3-cyclohexylpropanoic acid NA 840000 NA NA NA NA BindingDB
NMT1 (2S)-2-[[(2S)-6-amino-2-[[(2S)-3-hydroxy-2-[[2-[4-[4-(2-methylimidazol-1-yl)butyl]phenyl]acetyl]amino]propanoyl]amino]hexanoyl]amino]-3-cyclohexylpropanoic acid NA 809500 NA NA NA NA BindingDB
NMUR2 2-(2-Fluoro-5-methoxyphenyl)-3-hydroxychromen-4-one NA NA NA 253000 NA NA TTD
NOS1 Propargylguanidine 12000000 NA NA NA NA NA TTD
NOS1 7-(2-methoxyethoxy)-2-[2-(4-methoxypyridin-2-yl)ethyl]-1H-imidazo[4,5-b]pyridine NA 123026.88 NA NA NA NA BindingDB|TTD
NOS1 (1R)-1-Amino-4-{[(E)-amino(imino)methyl]amino}butylboronic acid NA 300000 NA NA NA NA BindingDB