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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
NMT1 4-[3-[[(2S)-4-methylmorpholin-2-yl]methoxy]propyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide NA 340000 NA NA NA NA BindingDB
NMT1 4-[3-(4-methylpiperazin-1-yl)propyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide NA 550000 NA NA NA NA BindingDB
NMT1 N-[6-(2-methylpropyl)quinolin-5-yl]-4-[3-[[(2S)-morpholin-2-yl]methoxy]propyl]benzenesulfonamide NA 390000 NA NA NA NA BindingDB
NMT1 N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-(1-methylpiperidin-4-yl)propyl]benzenesulfonamide NA 280000 NA NA NA NA BindingDB
NMT1 N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-[[(2R)-4-methylmorpholin-2-yl]methoxy]propyl]benzenesulfonamide NA 130000 NA NA NA NA BindingDB
NMT1 N-[6-(2-methylpropyl)quinolin-5-yl]-4-(4-piperidin-4-ylbutyl)benzenesulfonamide NA 240000 NA NA NA NA BindingDB
NMT1 4-[3-[(3R)-1-methylpiperidin-3-yl]oxypropyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide NA 1200000 NA NA NA NA BindingDB
NMT1 4-[4-(4-methyl-1,4-diazepan-1-yl)butyl]-N-[6-(2-methylpropyl)quinolin-5-yl]benzenesulfonamide NA 1400000 NA NA NA NA BindingDB
NMT1 N-[2-methyl-5-(2-methylpropyl)indazol-4-yl]-4-[3-[[(3S)-4-methylmorpholin-3-yl]methoxy]propyl]benzenesulfonamide NA 4600000 NA NA NA NA BindingDB
NMT1 4-Oxo-4-(phenylamino)isocrotonic acid NA 203000 NA NA NA NA BindingDB
NMT1 (Z)-4-(2,6-dimethylanilino)-4-oxobut-2-enoic acid NA 434000 NA NA NA NA BindingDB
NMT1 (Z)-methyl 4-(3,4-dichlorophenylamino)-4-oxobut-2-enoate NA 431600 NA NA NA NA BindingDB
NMT1 3-(3-Butyl-6-Methoxy-2-Methyl-Quinolin-4-Yl)sulfanylpropanenitrile NA 115000 NA NA NA NA BindingDB
NMT1 (2Z)-4-[(4-nitrophenyl)amino]-4-oxobut-2-enoic acid NA 246000 NA NA NA NA BindingDB
NMT1 Methyl N-(3,4-dimethylphenyl)fumaramate NA 2330000 NA NA NA NA BindingDB
NMT1 (2S)-6-amino-2-[[(2S)-2-[2-[4-[4-(2-chloroimidazol-1-yl)butyl]phenyl]propanoylamino]-3-hydroxy-propanoyl]amino]-N-(2-cyclohexylethyl)hexanamide NA 142000 NA NA NA NA BindingDB
NMT1 (2S)-6-amino-N-(2-cyclohexylethyl)-2-[[(2S)-3-hydroxy-2-[2-[4-[4-(2-methylbenzimidazol-1-yl)butyl]phenyl]propanoylamino]propanoyl]amino]hexanamide NA 119500 NA NA NA NA BindingDB
NMT1 Ethyl 4-[2-hydroxy-3-(isopropylamino)propoxy]-3-methyl-1-benzofuran-2-carboxylate NA 194000 NA NA NA NA BindingDB
NMT1 Ethyl 3-methyl-4-{3-[(methylethyl)amino]propoxy}benzo[d]furan-2-carboxylate NA 380000 NA NA NA NA BindingDB
NMT1 Ethyl 4-{3-[(tert-butyl)amino]-2-hydroxypropoxy}-3-methylbenzo[d]furan-2-carboxylate NA 470000 NA NA NA NA BindingDB