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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
NOS1 methyl (2S)-2-[[(E)-3-(3,4-dichlorophenyl)prop-2-enoyl]amino]-3-(4-fluorophenyl)propanoate NA 148510 NA NA NA NA BindingDB
NOS1 Aminoguanidine NA 118000 NA NA NA NA BindingDB|PubChem
NOS1 (2S)-2-amino-5-[carbamoyl(methyl)amino]pentanoic acid NA 7900000 NA NA NA NA BindingDB|TTD
NOS1 methyl (2S)-2-[[(E)-3-(3,4-dichlorophenyl)prop-2-enoyl]amino]-3-phenylpropanoate NA 110555 NA NA NA NA BindingDB
NOS1 1-(4-(2-bromophenoxy)butyl)-1H-imidazole 180000 NA NA NA NA NA BindingDB|TTD
NOS1 1-(3-(4-bromophenoxy)propyl)-1H-imidazole 125000 NA NA NA NA NA BindingDB|TTD
NOS1 NA 145000 NA NA NA NA BindingDB
NOS1 methyl (2S)-2-[[(E)-3-(4-chlorophenyl)prop-2-enoyl]amino]-3-phenylpropanoate NA 102382 NA NA NA NA BindingDB
NOS1 Amino(prop-2-ynylamino)methaniminium 12000000 NA NA NA NA NA BindingDB
NOS1 ((E)-3-But-2-enyl)-[1,4]oxazepan-(5Z)-ylideneamine NA 108000 NA NA NA NA BindingDB|TTD
NOS1 N-(2-Amino-6,7-diphenyl-pteridin-4-yl)-isobutyramide NA 192000 NA NA NA NA BindingDB|TTD
NOS1 2-Benzyloxycarbonylamino-3-phenyl-propionic acid 2,4-diamino-pteridin-6-ylmethyl ester NA 180000 NA NA NA NA BindingDB|TTD
NOS1 NA 111100 NA NA NA NA BindingDB
NOS1 NA 125000 NA NA NA NA BindingDB
NOS1 NA 130000 NA NA NA NA BindingDB
NOS1 NA 172000 NA NA NA NA BindingDB
NOS1 2,4-Diamino-7,8-dihydro-6H-pteridine-5-carbaldehyde NA 300000 NA NA NA NA BindingDB|TTD
NOS1 (S)-3-(2-Acetimidoylamino-ethanesulfonyl)-2-amino-propionic acid NA 630000 NA NA NA NA BindingDB|TTD
NOS1 NA 116900 NA NA NA NA BindingDB
NOS1 (R)-5-Acetimidoylamino-2-(S)-amino-3-methyl-pentanoic acid NA 1000000 NA NA NA NA TTD