| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| NOS1 |
2-[(4-Ethoxyphenyl)methyl]-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-nitrobenzimidazole;dihydrochloride |
NA |
113000 |
NA |
NA |
NA |
NA |
TTD |
| NOS1 |
(2S)-2-amino-5-[[(hydroxyamino)-nitrosomethyl]-methylamino]pentanoic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB |
| NOS1 |
1H-Indazole |
NA |
178000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS1 |
1H-Indazole, 3-chloro-6-nitro- |
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS1 |
3,5-Dimethylpyrazole-1-carboxamidine |
350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS1 |
L-Homocysteine, S-(2-((1-iminoethyl)amino)ethyl)- |
NA |
144543.98|145000|177000|144544 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| NOS1 |
N*4*,N*4*-Dibenzyl-6-phenyl-pteridine-2,4-diamine |
NA |
129300 |
NA |
NA |
NA |
NA |
BindingDB |
| NOS2 |
Saquayamycins A1 |
NA |
101200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
[(1R)-1-acetamido-4-(diaminomethylideneamino)butyl]boronic acid;hydrochloride |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| NOS2 |
[(1R)-1-amino-4-(diaminomethylideneamino)butyl]boronic acid;dihydrochloride |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
5-(3,5-Dihydroxyphenethyl)-1,3-benzenediol |
NA |
432600 |
NA |
NA |
NA |
NA |
BindingDB |
| NOS2 |
8-Fluoro-3-(4-fluoro-phenyl)-3,4-dihydro-isoquinolin-1-ylamine |
NA |
350000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
N*4*,N*4*-Dibenzyl-6-(4-methoxy-phenyl)-pteridine-2,4-diamine |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
6-(4-Chloro-phenyl)-4-piperidin-1-yl-5,6,7,8-tetrahydro-pteridin-2-ylamine |
NA |
106200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
6-(4-methoxyphenyl)-4-N,4-N-dipropyl-5,6,7,8-tetrahydropteridine-2,4-diamine |
NA |
280500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
3-Cyclopropyl-3,4-dihydro-isoquinolin-1-ylamine |
NA |
300000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
3-(3-fluorophenyl)-N-[2-[2-(4-methylimidazol-1-yl)pyrimidin-4-yl]ethyl]propan-1-amine |
287000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| NOS2 |
1-[3-(2-Amino-5-methoxyphenyl)-3-hydroxypropyl]-3-methylthiourea |
NA |
180000|130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| NOS2 |
1-[3-(2-Amino-5-chlorophenyl)-3-hydroxypropyl]-3-methylthiourea |
NA |
710000 |
NA |
NA |
NA |
NA |
TTD |
| NOS2 |
1-[3-(2-Aminophenyl)-3-hydroxypropyl]-3-methylthiourea |
NA |
350000 |
NA |
NA |
NA |
NA |
TTD |