| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDGFRB |
6-[5-[(1S)-1-amino-2-methylsulfonylethyl]furan-2-yl]-N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]quinazolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
6-[(2,4-dichlorophenyl)methyl]-4-N-(3-fluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
183100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
6-[(2,4-dichlorophenyl)methyl]-4-N-[3-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
6-[(2,4-dichlorophenyl)methyl]-4-N-(3-ethynylphenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
N4-(3-Fluoro-4-trifluoromethylphenyl)-6-(2,4-dichlorobenzyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
N4-(4-Isopropylphenyl)-6-(2,4-dichlorobenzyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
174900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
N-(3-bromophenyl)-6-(2-methylbenzyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
182000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
N-(3-bromophenyl)-6-(2,5-dimethoxybenzyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
171300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
N-(3-bromophenyl)-6-(2,4-dichlorobenzyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
220400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
6-(2,4-dichlorobenzyl)-N-(3-(trifluoromethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
110100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
6-(2,4-dichlorobenzyl)-N-(3-ethynylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
142200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
N-(3-ethynylphenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
6-(2-Phenylethyl)-N-[3-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
N-(3-bromo-4-fluorophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
192400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
N-[4-fluoro-3-(trifluoromethyl)phenyl]-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
N-(4-chloro-2-fluorophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
N-1H-indol-5-yl-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
104200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDGFRB |
2-Amino-4-(N-methyl-m-bromoanilino)-6-(2-methylbenzyl)-7-methyl-pyrrolo[2,3-d]pyrimidine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
2-Amino-4-(N-methyl-m-bromoanilino)-6-(2,5-dimethoxybenzyl)-7-methyl-pyrrolo[2,3-d]pyrimidine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PDGFRB |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |