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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PDE8A Roflumilast NA 200000 NA NA NA NA PubChem
PDE8A Rolipram NA 200000 NA NA NA NA PubChem
PDE8A Zardaverine NA 160000 NA NA NA NA BindingDB
PDE8A Filaminast NA 120000 NA NA NA NA BindingDB
PDE9A Tadalafil NA 150000 NA NA NA NA BindingDB
PDE9A 6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide NA 200000 NA NA NA NA TTD
PDE9A 6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide NA 200000 NA NA NA NA TTD
PDE9A Isobutylmethylxanthine NA 117000 NA NA NA NA TTD
PDF N-(1-benzenesulfonyl-5-bromo-2-methyl-1H-indol-3-ylmethyl)-N-hydroxyformamide NA 200000 NA NA NA NA BindingDB|TTD
PDF 1-(5-bromo-1H-indol-3-yl)-3-(hydroxyamino)propan-2-one NA 360000 NA NA NA NA BindingDB|TTD
PDF 1-(4-fluoro-1H-indol-3-yl)-3-(hydroxyamino)propan-2-one NA 700000 NA NA NA NA BindingDB|TTD
PDF 1-(5-chloro-1H-indol-3-yl)-3-(hydroxyamino)propan-2-one NA 600000 NA NA NA NA BindingDB|TTD
PDF 1-(6-bromo-1H-indol-3-yl)-3-(hydroxyamino)propan-2-one NA 250000 NA NA NA NA BindingDB|TTD
PDF 2-(5-bromo-2-methyl-1H-indolyl)-N-hydroxyacetamide NA 450000 NA NA NA NA BindingDB|TTD
PDGFRB N4-(3-bromo-4-fluorophenyl)-6-phenethyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine NA 500000 NA NA NA NA TTD
PDGFRB 5-[(1z)-2-(2-Methoxyphenyl)prop-1-En-1-Yl]furo[2,3-D]pyrimidine-2,4-Diamine NA 151900 NA NA NA NA TTD
PDGFRB N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[1-(cyclohexylamino)-2-methylsulfonylethyl]furan-2-yl]quinazolin-4-amine NA 200000 NA NA NA NA TTD
PDGFRB N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[2-methylsulfonyl-1-(propan-2-ylamino)ethyl]furan-2-yl]quinazolin-4-amine NA 200000 NA NA NA NA TTD
PDGFRB N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[2-methylsulfonyl-1-(2-methylsulfonylethylamino)ethyl]furan-2-yl]quinazolin-4-amine NA 200000 NA NA NA NA TTD
PDGFRB [[(1S)-1-[5-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-yl]-2-methylsulfonylethyl]amino] propanoate NA 200000 NA NA NA NA TTD