| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE7A |
N-(3-chlorophenyl)-2-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
4-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)-N-(4-propan-2-ylphenyl)butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
2-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)-N-(4-propan-2-ylphenyl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(4-butan-2-ylphenyl)-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide;hydrochloride |
NA |
125500 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE7A |
1-cyclopentyl-2-(furan-2-yl)-N-(2-methoxyethyl)imidazo[4,5-c]pyridin-4-amine |
NA |
191510 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE7A |
3-cyclopentyl-2-(furan-2-yl)-N-(2-methoxyethyl)imidazo[4,5-b]pyridin-7-amine |
NA |
118600 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE7A |
5-[4-(2-methoxyphenyl)piperazin-1-yl]-N-(4-propan-2-ylphenyl)pentanamide;hydrochloride |
NA |
151300 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE7A |
1-cyclopentyl-2-(furan-2-yl)-N-(3-methoxypropyl)imidazo[4,5-c]pyridin-4-amine |
NA |
142390 |
NA |
NA |
NA |
NA |
BindingDB |
| PDE7A |
Theophylline |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE7A |
Crisaborole |
NA |
2030000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PDE7A |
Rolipram |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PDE7B |
Roflumilast |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE7B |
Rolipram |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE8A |
Tadalafil |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE8A |
Sildenafil |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PDE8A |
6-cyclopentyloxy-7-methoxy-1-phenyl-N-[2-(trifluoromethoxy)phenyl]-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE8A |
6-cyclopentyloxy-7-methoxy-N-(2-methoxyphenyl)-1-phenyl-3,4-dihydroisoquinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE8A |
Isobutylmethylxanthine |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |