| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDE7A |
HC-030031 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
5-Chloro-2-(2-nitrophenyl)sulfanylaniline |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE7A |
4-(1,3-dimethyl-2,6-dioxopurin-7-yl)-N-[(E)-(2-hydroxyphenyl)methylideneamino]butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-[(E)-(2,4-dihydroxyphenyl)methylideneamino]-4-(1,3-dimethyl-2,6-dioxopurin-7-yl)butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
4-[1,3-dimethyl-2,6-dioxo-8-(pyridin-2-ylmethylamino)purin-7-yl]-N-[(E)-(2-hydroxyphenyl)methylideneamino]butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-[(E)-(2,4-dihydroxyphenyl)methylideneamino]-4-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)butanamide |
NA |
140900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE7A |
4-[8-(furan-2-ylmethylamino)-1,3-dimethyl-2,6-dioxopurin-7-yl]-N-[(E)-(2-hydroxyphenyl)methylideneamino]butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
4-[8-(benzylamino)-1,3-dimethyl-2,6-dioxopurin-7-yl]-N-[(E)-(2,4-dihydroxyphenyl)methylideneamino]butanamide |
NA |
115900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDE7A |
4-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)-N-[(E)-(2-hydroxy-4-methoxyphenyl)methylideneamino]butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
4-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)-N-[(E)-(2-methoxyphenyl)methylideneamino]butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-[(2-chlorophenyl)methyl]-2-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(3-chlorophenyl)-2-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-[(2-chlorophenyl)methyl]-2-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(4-tert-butylphenyl)-2-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(3-chlorophenyl)-4-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(4-tert-butylphenyl)-2-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(4-chlorophenyl)-4-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-(4-chlorophenyl)-2-(8-ethoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
2-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)-N-(4-propan-2-ylphenyl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PDE7A |
N-[(2-chlorophenyl)methyl]-4-(8-methoxy-1,3-dimethyl-2,6-dioxopurin-7-yl)butanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |