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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PHF8 N-(Carboxycarbonyl)-S-(Naphthalen-2-Ylmethyl)-L-Cysteine NA 1000000 NA NA NA NA TTD
PHF8 (2R)-3-(naphthalen-1-ylmethylsulfanyl)-2-(oxaloamino)propanoic acid NA 1000000 NA NA NA NA TTD
PHF8 2-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]ethyl-trimethylazanium;iodide NA 307000 NA NA NA NA TTD
PHF8 3-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]propyl-trimethylazanium;iodide NA 390000 NA NA NA NA TTD
PHF8 Methyl 3-[hydroxy(10-methylundecanoyl)amino]propanoate NA 150000 NA NA NA NA TTD
PHGDH 1-(2-Bromophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone NA 160700 NA NA NA NA TTD
PHGDH 1-(3-Fluorophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone NA 200000 NA NA NA NA TTD
PHGDH 2-Morpholin-4-yl-1-(2-nitrophenyl)-2-sulfanylideneethanone NA 200000 NA NA NA NA TTD
PHGDH 1-(3-Bromophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone NA 200000 NA NA NA NA TTD
PHGDH 1-(2-Fluorophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone NA 200000 NA NA NA NA TTD
PHGDH 1-([1,1'-Biphenyl]-4-yl)-2-morpholino-2-thioxoethan-1-one NA 200000 NA NA NA NA TTD
PHGDH 1-(3-Iodophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone NA 200000 NA NA NA NA TTD
PHGDH 1-(2-Iodophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone NA 200000 NA NA NA NA TTD
PHGDH 4-[3-[(4,5-Dichloro-1-methylindol-2-yl)methylamino]oxetan-3-yl]benzoic acid NA 209000 NA NA NA NA TTD
PHPT1 Ethacrynic Acid 183000 NA NA NA NA NA PubChem
PHPT1 Ethylmaleimide 209000 NA NA NA NA NA PubChem
PI4K2A Adenosine-5'-diphosphate 100100|NA NA|145300 NA NA NA NA PubChem
PI4K2B Adenosine-5'-diphosphate NA|100100 145300|NA NA NA NA NA PubChem
PI4KA Adenosine-5'-diphosphate 100100|NA NA|145300 NA NA NA NA PubChem
PI4KB Adenosine-5'-diphosphate 100100|NA NA|145300 NA NA NA NA PubChem