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negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
PGR
Aztreonam
NA
NA
NA
NA
NA
400000
PubChem
PGR
Carumonam
NA
NA
NA
NA
NA
500000|320000
PubChem
PGR
Doripenem
NA
NA
NA
NA
NA
300000
PubChem
PGR
Miristalkonium chloride
NA
NA
NA
NA
22387200
NA
PubChem
PHF8
2,4-Pyridinedicarboxylic acid
NA
250000
NA
NA
NA
NA
TTD
PHF8
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-difluorophenoxy]propyl-trimethylazanium;iodide
NA
242000
NA
NA
NA
NA
TTD
PHF8
3-[2-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-trimethylazanium;iodide
NA
496000
NA
NA
NA
NA
TTD
PHF8
Trimethyl-[3-[4-(2-methyl-1-benzofuran-3-carbonyl)phenoxy]propyl]azanium;iodide
NA
126000
NA
NA
NA
NA
TTD
PHF8
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-trimethylazanium;iodide
NA
355000
NA
NA
NA
NA
TTD
PHF8
(2-Butyl-1-benzofuran-3-yl)-[4-[3-(dimethylamino)propoxy]phenyl]methanone
NA
397000
NA
NA
NA
NA
TTD
PHF8
Trimethyl-[3-[2-(2-methyl-1-benzofuran-3-carbonyl)phenoxy]propyl]azanium;iodide
NA
286000
NA
NA
NA
NA
TTD
PHF8
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-dimethoxyphenoxy]propyl-trimethylazanium;iodide
NA
240000
NA
NA
NA
NA
TTD
PHF8
[4-(3-Aminopropoxy)phenyl]-(2-butyl-1-benzofuran-3-yl)methanone
NA
386000
NA
NA
NA
NA
TTD
PHF8
Trimethyl-[3-[4-(2-methyl-1-benzothiophene-3-carbonyl)phenoxy]propyl]azanium;iodide
NA
377000
NA
NA
NA
NA
TTD
PHF8
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-triethylazanium;iodide
NA
221000
NA
NA
NA
NA
TTD
PHF8
3-[4-[C-(1-benzofuran-3-yl)-N-methylcarbonimidoyl]phenoxy]propyl-trimethylazanium;iodide
NA
697000
NA
NA
NA
NA
TTD
PHF8
Amiodarone
NA
252000
NA
NA
NA
NA
PubChem|TTD
PHF8
N'1,N'1,N'4,N'4-Tetramethylsuccinohydrazide
NA
117000
NA
NA
NA
NA
TTD
PHF8
Oxalylglycine
NA
250000
NA
NA
NA
NA
TTD
PHF8
N-(Carboxycarbonyl)-S-(3-Nitrobenzyl)-L-Cysteine
NA
1000000
NA
NA
NA
NA
TTD
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