| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PEPD |
2-((1R,2R)-2-Carboxy-cyclohexyl)-2-oxo-ethyl-ammonium; chloride |
1100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PEX5L |
US20230391714, Nucc-0201100 |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| PEX5L |
US20230391714, Nucc-0201101 |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| PEX5L |
US20230391714, Nucc-0201182 |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| PEX5L |
US20230391714, Nucc-0201228 |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| PFKFB3 |
3H-benzo[e]indol-2-yl(pyridin-4-yl)methanone |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
4-bromo-5-(morpholin-4-yl)-2-phenylpyridazin-3(2H)-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
2-(5-bromo-6-oxo-1-phenylpyridazin-4-yl)-3,4-dihydro-1H-isoquinoline-5-carbonitrile |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
4-Bromo-5-(2-oxa-6-azaspiro[3.3]heptan-6-yl)-2-phenylpyridazin-3-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
5-(4-Acetyl-5-methyltriazol-1-yl)-2-phenyl-4-propan-2-ylpyridazin-3-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
5-(4-Acetyl-5-methyltriazol-1-yl)-4-bromo-2-[[4-[2-(dimethylamino)ethylamino]phenyl]methyl]pyridazin-3-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
2-[(5-Bromo-6-oxo-1-phenylpyridazin-4-yl)amino]acetamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
5-(4-Acetyl-5-methyltriazol-1-yl)-4-ethoxy-2-phenylpyridazin-3-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
4-Bromo-5-(oxolan-2-ylmethylamino)-2-phenylpyridazin-3-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PFKFB3 |
5-(4-Acetyl-5-methyltriazol-1-yl)-2-benzylpyridazin-3-one |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PGA5 |
2-Benzyl-N-[1-(1-cyclohexylmethyl-2,3,4,5,6-pentahydroxy-hexylcarbamoyl)-2-(1H-imidazol-4-yl)-ethyl]-3-(2-methyl-propane-2-sulfonyl)-propionamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PGA5 |
(S)-N-[(S)-2-(2-Amino-thiazol-4-yl)-1-((1S,2R,3S)-1-cyclohexylmethyl-2,3-dihydroxy-5-methyl-hexylcarbamoyl)-ethyl]-2-(morpholine-4-sulfonylamino)-3-phenyl-propionamide |
NA |
202000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PGD |
[(4R,5R)-5-carbamoyl-2,2-dimethyl-1,3-dioxolan-4-yl]methyl dihydrogen phosphate |
588000|714000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PGD |
((R)-2-Hydroxy-3-phosphonooxy-propane-1-sulfinyl)-acetic acid |
198000|784000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PGD |
((R)-2-Acetoxy-3-phosphonooxy-propane-1-sulfinyl)-acetic acid |
625000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |