Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| PDPK1 | 4-Bromo-3-chloro-2H-indazole | NA | 163600 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| PDPK1 | [(S)-phenyl-[[(2R)-2-phenylpropyl]amino]methyl]phosphonic acid | NA | NA | 150000 | NA | NA | NA | BindingDB |
| PDPK1 | Acetic acid, 2-[[3-(4-chlorophenyl)-3-oxo-1-phenylpropyl]thio]- | NA | NA | NA | 133000 | NA | NA | BindingDB|TTD |
| PDPK1 | NA | 492000 | NA | NA | NA | NA | BindingDB | |
| PDPK1 | NA | 461000 | NA | NA | NA | NA | BindingDB | |
| PDPK1 | NA | 122000 | NA | NA | NA | NA | BindingDB | |
| PDPK1 | Isoquinolin-3-Amine | NA | 376000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| PDPK1 | 5,6-dimethyl-3H,4H-thieno(2,3-d)pyrimidin-4-one | NA | 828000 | NA | NA | NA | NA | BindingDB|TTD |
| PDPK1 | 2-(3-anilino-2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl)acetic acid | NA | NA | NA | 900000 | NA | NA | BindingDB|TTD |
| PDPK1 | 2-(2-oxo-3-phenylsulfanyl-4,5-dihydro-3H-1-benzazepin-1-yl)acetic acid | NA | NA | NA | 101000 | NA | NA | BindingDB|TTD |
| PDPK1 | 4-(1-(carboxymethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-ylthio)benzoic acid | NA | NA | NA | 187000 | NA | NA | BindingDB|TTD |
| PDPK1 | 3-(furan-2-yl)-1H-pyrazol-5-amine | NA | 313000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| PDPK1 | 3,5-Diamino-1,2,4-triazine-6-carboxamide | NA | 145000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| PDPK1 | US8628961, Pit-3 | NA | 106800 | NA | NA | NA | NA | BindingDB |
| PDPK1 | 4-amino-1H-pyrazole-5-carboxamide | NA | 200000|2e+05 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| PDPK1 | NA | 345000 | NA | NA | NA | NA | BindingDB | |
| PDPK1 | 4-[(3,4,5-Trifluorophenyl)methylamino]quinazoline-8-carboxamide | NA | 102000 | NA | NA | NA | NA | BindingDB |
| PDPK1 | 6-Methoxypurine | NA | 340000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| PDPK1 | NA | 106000 | NA | NA | NA | NA | BindingDB | |
| PDPK1 | NA | 154000 | NA | NA | NA | NA | BindingDB |