| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDK4 |
Dichloroacetic Acid |
NA |
2000000|727000 |
NA |
NA |
NA |
NA |
PubChem |
| PDK4 |
Nandrolone |
NA |
120000 |
NA |
NA |
NA |
NA |
PubChem |
| PDPK1 |
3-(hydroxymethyl)-1H-pyrazol-5-ol |
NA |
344000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
7-chlorothieno[3,2-b]pyridin-5(4H)-one |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
1H-indazol-3-amine |
NA |
311000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
4-Hydroxyquinazoline |
NA |
345000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PDPK1 |
3H,4H-thieno[3,2-d]pyrimidin-4-one |
NA |
492000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one |
NA |
461000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
6-(4-fluorophenyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one |
NA |
122000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
Imidazo[4,5-d]pyridazin-4-one, 7-methyl-1,5-dihydro- |
NA |
472000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
7-(Methylamino)thieno[3,2-d]pyrimidin-4(3H)-one |
NA |
154000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
7-(dimethylamino)-3H-thieno[3,2-d]pyrimidin-4-one |
NA |
109000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
6-(4-fluorophenyl)-7-methyl-3H-thieno[3,2-d]pyrimidin-4-one |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
| PDPK1 |
3,4-dihydroisoquinolin-1(2H)-one |
NA |
169000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
4-(1H-pyrazol-3-yl)pyridine |
NA |
326000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
7,8,9,10-tetrahydropyrazino[1,2-b]indazol-1(2H)-one |
NA |
273000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDPK1 |
2-{2-[2-(2,3-Dimethylphenoxy)ethylthio]benzimidazolyl}acetic acid |
NA |
NA |
110000 |
NA |
NA |
NA |
BindingDB |
| PDPK1 |
5-Fluoroindole-2-carboxylic acid |
NA |
297000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDPK1 |
5H,6H,7H,8H-(1,2,4)triazolo(4,3-a)pyridine |
NA |
244000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
2-Amino-4-hydroxybenzothiazole |
NA |
256000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |