| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PDPK1 |
|
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDPK1 |
{[1-(2-Phenoxyethyl)-1H-benzimidazol-2-yl]-thio}acetic acid |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| PDPK1 |
{2-[(1-naphthylmethyl)thio]-1H-benzimidazol-1-yl}acetic acid |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| PDPK1 |
3-Amino-5-bromo-1H-indazole |
NA |
101900 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
3-Amino-1,2,4-benzotriazine |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PDPK1 |
3,4-dimethyl-2,3-dihydro-1H-pyrano[2,3-c]pyrazol-6-one |
NA |
302000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDPK1 |
|
NA |
472000 |
NA |
NA |
NA |
NA |
BindingDB |
| PDPK1 |
N-(6-fluoro-1,3-benzothiazol-2-yl)acetamide |
NA |
402000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PDXK |
4-Ethynyl-5-(hydroxymethyl)-2-methylpyridin-3-ol |
125000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PDXK |
2-Ethynyl-4,5-bis(hydroxymethyl)pyridin-3-ol |
105000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PEPD |
H-Sta(3R,4S)-Pro-Ala-NH2 |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| PEPD |
H-bAla(2S-OH,3R-Bn)-Hyp-Pro-Ala-NH2 |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| PEPD |
2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolidin-1-yl]-4-phenyl-butyric acid |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| PEPD |
H-bAla(2R-OH,3R-iBu)-Pro-Ala-NH2 |
NA |
410000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PEPD |
Aminolevulinic Acid |
960000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PEPD |
(2S)-N-[(2S)-1-amino-1-oxopropan-2-yl]-1-[2-(hydroxycarbamoyl)cyclohexanecarbonyl]pyrrolidine-2-carboxamide |
NA |
1700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PEPD |
(2S)-N-[(2S)-1-amino-1-oxopropan-2-yl]-1-(2-sulfanylcyclopentanecarbonyl)pyrrolidine-2-carboxamide |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| PEPD |
1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydroxy-pyrrolidine-2-carbonyl]-pyrrolidine-2-carboxylic acid (1-carbamoyl-ethyl)-amide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| PEPD |
H-bAla(2S-OH,3R-Bn)-Pro-Pro-Ala-Ala-Cys-NH2 |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PEPD |
(1R,2R)-2-(2-aminoacetyl)cyclohexane-1-carboxylic acid;hydrochloride |
1100000 |
NA |
NA |
NA |
NA |
NA |
TTD |