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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PDGFRB N-[5-chloro-4-(3-methoxyanilino)-9H-pyrimido[4,5-b]indol-2-yl]-2,2-dimethylpropanamide NA 196200 NA NA NA NA BindingDB|TTD
PDGFRB 4-N-(3-bromophenyl)-1H-indeno[2,1-d]pyrimidine-2,4-diamine NA 126300 NA NA NA NA BindingDB
PDK1 (1E,4S,4aR,5R,6aS,7S,9aR)-5-(acetyloxy)-1-[[[3-(dimethylamino)propyl]methylamino]methylene]-4a,5,6,6a,7,8,9,9a-octahydro-cyclopenta[5,6]naphtho[1,2-c]pyran-2,10(1H,4H)-dione NA 200000 NA NA NA NA TTD
PDK1 [(1S,3aR,6E,9S,9aR,10R,11aS)-6-[[tert-butyl(2-hydroxyethyl)amino]methylidene]-1,5-dihydroxy-9-(methoxymethyl)-9a,11a-dimethyl-4,7-dioxo-2,3,3a,9,10,11-hexahydro-1H-indeno[4,5-h]isochromen-10-yl] acetate NA 200000 NA NA NA NA TTD
PDK1 Sodium Dichloroacetate NA 1000000|NA NA|1000000 NA|130000|5700000 NA NA PubChem|TTD
PDK1 Monorden NA 230000 NA NA NA NA TTD
PDK1 Dichloroacetic Acid NA 2000000|1025000|5100000 NA NA NA NA PubChem|TTD
PDK1 4-[4-(4-methoxyphenyl)-5-methyl-1H-pyrazol-3-yl]benzene-1,3-diol NA 648000 NA NA NA NA TTD
PDK1 Nandrolone NA 120000 NA NA NA NA PubChem
PDK2 Methyl 2,4-Dihydroxybenzoate NA 192000 NA NA NA NA ChEMBL
PDK2 Sodium Dichloroacetate NA NA|1000000 NA 130000|NA NA NA PubChem
PDK2 Dichloroacetic Acid NA 2000000|9000000|504000 NA NA NA NA PubChem|TTD
PDK2 Nandrolone NA 120000 NA NA NA NA PubChem
PDK3 Sodium Dichloroacetate NA NA|1000000 NA 130000|NA NA NA PubChem
PDK3 Monorden NA 230000 NA NA NA NA TTD
PDK3 Dichloroacetic Acid NA 2000000|5560000 NA NA NA NA PubChem|TTD
PDK3 Nandrolone NA 120000 NA NA NA NA PubChem
PDK4 Methyl 2,4-Dihydroxybenzoate NA 345000 NA NA NA NA ChEMBL
PDK4 3,3-Dimethyl-1,3-dihydro-indol-2-one NA 890000 NA NA NA NA ChEMBL
PDK4 Sodium Dichloroacetate NA 1000000|NA NA NA|130000 NA NA PubChem