| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIK3CB |
3-(4-Morpholino-1-methyl-1H-pyrazolo[3,4-d]pyrimidine-6-yl)phenol |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide |
NA |
50118723 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-propylpyridine-3-sulfonamide |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-propan-2-ylpyridine-3-sulfonamide |
NA |
63095734|63095734.45 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N,N-diethylpyridine-3-sulfonamide |
NA |
25118864|25118864.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-methylpyridine-3-sulfonamide |
NA |
39810717|39810717.06 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-(2,2,2-trifluoroethyl)pyridine-3-sulfonamide |
NA |
12589254|12589254.12 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
CID 44621449 |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-phenylpyridine-3-sulfonamide |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-benzylpyridine-3-sulfonamide |
NA |
25118864|25118864.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
7-(5-Methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine |
NA |
39810717|39810717.06 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)pyridine-3-sulfonamide |
NA |
39810717|39810717.06 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
5-(2-amino-5-fluoro-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
4-(1-(7-Fluoro-3-methyl-2-(2-pyridinyl)-4-quinolinyl)-3,3-dimethyl-2,3-dihydro-1H-indol-6-yl)-6-methyl-2-pyrimidinamine |
125000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PIK3CB |
N-[7-methyl-6-(5-methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]acetamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
7-[5-(2,2-Dimethylazetidin-1-yl)sulfonylpyridin-3-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine |
NA |
50118723|50118723.36 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CB |
4-N-benzyl-6-morpholin-4-ylpyrimidine-2,4-diamine |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PIK3CB |
N-benzyl-4-methyl-6-morpholin-4-ylpyrimidin-2-amine |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PIK3CB |
4-(2-Amino-1,3-benzothiazol-6-yl)-1-(cyclopropylmethyl)pyridin-2-one |
NA |
125892.54 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CB |
IC-87114 |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |