| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIK3CD |
13-Morpholin-4-yl-11-(morpholin-4-ylmethyl)-8-phenyl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
13-Morpholin-4-yl-11-(1-morpholin-4-ylethyl)-8-phenyl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
154780 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
4-(2-Amino-1,3-benzothiazol-6-yl)-1-(2-methoxyethoxy)pyridin-2-one |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CD |
1-(cyclopropylmethyl)-4-[2-[[(1R)-1-(oxan-4-yl)ethyl]amino]-1,3-benzothiazol-6-yl]pyridin-2-one |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CD |
1-(cyclopropylmethyl)-4-[2-[[(1S)-1-(oxan-4-yl)ethyl]amino]-1,3-benzothiazol-6-yl]pyridin-2-one |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CD |
1-(Cyclopropylmethyl)-4-[2-[(1,1-dioxothian-4-yl)methylamino]-1,3-benzothiazol-6-yl]pyridin-2-one |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CD |
4-[[5-(1H-indazol-4-yl)-1,3,4-oxadiazol-2-yl]methyl]morpholine |
NA |
158489|158489.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
1-[3-[4-(Dimethylamino)piperidine-1-carbonyl]phenyl]-3-[4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)phenyl]urea |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CD |
methyl (2Z)-2-[(2Z)-4-oxo-3-phenyl-2-[(E)-[4-(2,2,2-trifluoroethoxy)phenyl]methylidenehydrazinylidene]-1,3-thiazolidin-5-ylidene]acetate |
NA |
121300 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide |
NA |
50118723 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-propan-2-ylpyridine-3-sulfonamide |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N,N-diethylpyridine-3-sulfonamide |
NA |
12589254|12589254.12 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-methylpyridine-3-sulfonamide |
NA |
25118864|25118864.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-(2,2,2-trifluoroethyl)pyridine-3-sulfonamide |
NA |
7943282|7943282.35 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
CID 44621449 |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-phenylpyridine-3-sulfonamide |
NA |
25118864|25118864.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-benzylpyridine-3-sulfonamide |
NA |
19952623|19952623.15 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
7-(5-Methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine |
NA |
39810717|39810717.06 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)pyridine-3-sulfonamide |
NA |
31622777|31622776.6 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CD |
5-(2-amino-5-fluoro-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide |
NA |
7943282|7943282.35 |
NA |
NA |
NA |
NA |
BindingDB|TTD |