| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIN1 |
4-(benzylcarbamoyl)-2-phenyl-1H-imidazole-5-carboxylic acid |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIN1 |
Cycloheximide |
200000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PIN1 |
Procodazole |
NA |
740000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIN1 |
3-(2-Pyridinyl)-1H-pyrazole-5-carboxylic acid |
NA |
720000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIN1 |
5-(2-Methoxyphenyl)-2-furoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PIN4 |
Cycloheximide |
187000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PIPOX |
6-Oxa-3-azabicyclo[3.1.0]hexane-2-carboxylic acid, (1R,2S,5S)- |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIPOX |
(4S)-1,3-thiazinane-4-carboxylic acid |
36000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PIPOX |
(S)-pipecolate |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PITRM1 |
2-[4,7-bis(carboxymethyl)-10-[2-[[2-[[2-[[(2S)-1-[[(2R)-1-[(2S)-2-cyano-4,4-difluoropyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-2-oxoethyl]-1,4,7,10-tetrazacyclododec-1-yl]acetic acid |
NA |
157000 |
NA |
NA |
NA |
NA |
BindingDB |
| PKD2L1 |
Amiloride |
NA |
143000 |
NA |
NA |
NA |
NA |
GtoPDB |
| PKM |
7,11b-dihydrobenz(b)indeno(1,2-d)pyran-3,4,6a,9,10(6H)-pentol |
NA |
340000 |
NA |
NA |
NA |
NA |
PubChem |
| PKM |
Menadione |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |
| PKM |
Hematoxylin |
NA |
340000 |
NA |
NA |
NA |
NA |
PubChem |
| PKM |
Polydatin |
NA |
128000 |
NA |
NA |
NA |
NA |
PubChem |
| PKM |
Serine |
NA |
NA |
NA |
1300000 |
NA |
NA |
PubChem |
| PKN1 |
2-pyrimidin-5-yl-1H-benzimidazole-4-carboxamide |
NA |
137920 |
NA |
NA |
NA |
NA |
BindingDB |
| PKN1 |
5-Nitro-2-(4-pyridinyl)-1H-benzimidazole |
NA |
109300 |
NA |
NA |
NA |
NA |
BindingDB |
| PLA2G10 |
2-(1-Benzyl-6-methoxy-2-methyl-1H-indol-3-yl)-2-hydroxy-acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLA2G10BP |
2-(1-Benzyl-6-methoxy-2-methyl-1H-indol-3-yl)-2-hydroxy-acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
ChEMBL |