| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLA2G15 |
Ester Of Phospholipid |
NA |
9750000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLA2G1B |
4-[5-[[5-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-2,4-dimethoxy-3,6-dimethylphenyl]methyl]-2,4-dimethoxy-3,6-dimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
90000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
4-[4-[5-[3-[4-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-3-methoxy-2,5,6-trimethylphenoxy]carbonyl-4-methoxyphenyl]sulfonyl-2-methoxybenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
9000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
Bis[3-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-4-methoxyphenyl]ether |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
Bis[3-[[4-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-4-methoxyphenyl]sulfide |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
Bis[3-[[4-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-3-methoxy-2,5,6-triimethylphenoxy]carbonyl]-4-methoxyphenyl]sulfoxide |
NA |
11000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
Thielocin A1 |
NA |
135000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
4-[4-[2,4-Dihydroxy-3,6-dimethyl-5-[[(2-oxo-2-phenylmethoxyethyl)amino]methyl]benzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
4-[4-[2,4-dihydroxy-3,6-dimethyl-5-[[[(1S)-1-phenylethyl]amino]methyl]benzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoic acid |
NA |
60000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
4-[4-[5-[(2,4-Dimethoxy-3,6-dimethylphenyl)methyl]-2,4-dimethoxy-3,6-dimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
Thielocin-B3 |
NA |
18000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
Bis[3-[[4-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-3-methoxy-2,5,6-triimethylphenoxy]carbonyl]-4-methoxyphenyl]sulphide |
NA |
55000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
4-[4-[5-[3-[4-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-3-methoxy-2,5,6-trimethylphenoxy]carbonyl-4-methoxyphenoxy]-2-methoxybenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
6500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
4-[4-[5-[[5-[4-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-3-methoxy-2,5,6-trimethylphenoxy]carbonyl-2,4-dimethoxy-3,6-dimethylphenyl]methyl]-2,4-dimethoxy-3,6-dimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
4-[4-[5-[[5-[4-(4-Carboxy-3-hydroxy-2,5,6-trimethylphenoxy)carbonyl-3-hydroxy-2,5,6-trimethylphenoxy]carbonyl-2,4-dihydroxy-3,6-dimethylphenyl]methyl]-2,4-dihydroxy-3,6-dimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoic acid |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G1B |
4-[4-[5-[3-[4-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-3-methoxy-2,5,6-trimethylphenoxy]carbonyl-4-methoxy-5-methylphenoxy]-2,4-dimethoxybenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
6600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
Cholic Acid |
NA |
NA |
150000 |
NA |
NA |
NA |
PubChem |
| PLA2G1B |
4-(3-Benzyl-1-carbamoylmethyl-2-methyl-2,3-dihydro-indolizin-8-yloxy)-butyric acid methyl ester |
NA |
15000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
(3-Benzyl-1-carbamoylmethyl-2-methyl-2,3-dihydro-indolizin-8-yloxy)-acetic acid |
NA |
12000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G1B |
2-[[(3Z)-1-(2-amino-2-oxoethyl)-2-ethyl-3-(naphthalen-2-ylmethylidene)-2H-indolizin-8-yl]oxy]acetic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |