| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLA2G2A |
3-(Benzyl-hydroxy-amino)-1-(4-fluoro-phenyl)-propenone |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
3-(Benzyl-methoxy-amino)-1-(4-fluoro-phenyl)-propenone |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
4-[5-[[5-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-2,4-dimethoxy-3,6-dimethylphenyl]methyl]-2,4-dimethoxy-3,6-dimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
2800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
2-(1-Benzyl-5-methoxy-2-methyl-1H-indol-3-yl)-N-methyl-acetamide |
NA |
141800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
3-(1-Benzyl-3-carbamoylmethyl-2-ethyl-1H-indol-5-yloxy)-propane-1-sulfonic acid |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLA2G2A |
Bis[3-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-4-methoxyphenyl]ether |
NA |
75000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
2-(1-Benzyl-5-methoxy-2-methyl-1H-indol-3-yl)-octanoic acid hydrazide |
NA |
101200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
3-(1-Benzyl-3-carbamoylmethyl-2-methyl-1H-indol-5-yloxy)-benzoic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
2-(1-Benzyl-6-methoxy-2-methyl-1H-indol-3-yl)-2-hydroxy-acetamide |
NA |
120900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
Bis[3-[[4-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-4-methoxyphenyl]sulfide |
NA |
4800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
Bis[3-[[4-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-3-methoxy-2,5,6-triimethylphenoxy]carbonyl]-4-methoxyphenyl]sulfoxide |
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
Thielocin A1 |
NA |
12000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
4-[4-[2,4-Dihydroxy-3,6-dimethyl-5-[[(2-oxo-2-phenylmethoxyethyl)amino]methyl]benzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoic acid |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
4-[4-[2,4-dihydroxy-3,6-dimethyl-5-[[[(1S)-1-phenylethyl]amino]methyl]benzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoic acid |
NA |
840000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
4-[4-[5-[(2,4-Dimethoxy-3,6-dimethylphenyl)methyl]-2,4-dimethoxy-3,6-dimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
Bis[3-[[4-[(4-carboxy-3-methoxy-2,5,6-trimethylphenoxy)-carbonyl]-3-methoxy-2,5,6-triimethylphenoxy]carbonyl]-4-methoxyphenyl]sulphide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
4-[4-[5-[[5-[4-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-3-methoxy-2,5,6-trimethylphenoxy]carbonyl-2,4-dimethoxy-3,6-dimethylphenyl]methyl]-2,4-dimethoxy-3,6-dimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
4-[4-[5-[[5-[4-(4-Carboxy-3-hydroxy-2,5,6-trimethylphenoxy)carbonyl-3-hydroxy-2,5,6-trimethylphenoxy]carbonyl-2,4-dihydroxy-3,6-dimethylphenyl]methyl]-2,4-dihydroxy-3,6-dimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoyl]oxy-2-hydroxy-3,5,6-trimethylbenzoic acid |
NA |
2400000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G2A |
4-[4-[5-[3-[4-(4-Carboxy-3-methoxy-2,5,6-trimethylphenoxy)carbonyl-3-methoxy-2,5,6-trimethylphenoxy]carbonyl-4-methoxy-5-methylphenoxy]-2,4-dimethoxybenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoyl]oxy-2-methoxy-3,5,6-trimethylbenzoic acid |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G2A |
Quinacrine |
NA |
76000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |