| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLA2G2A |
3-(Cyclohexyl-hydroxy-amino)-1-(4-fluoro-phenyl)-propenone |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G3 |
Mitoxantrone |
NA |
121794 |
NA |
NA |
NA |
NA |
PubChem |
| PLA2G4A |
3-[2-[5-chloro-1-(diphenylmethyl)-2-methyl-1H-indol-3-yl]-ethoxy]benzoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G4A |
[5-chloro-1-(diphenylmethyl)-2-methyl-1H-indol-3-yl]acetic acid |
NA |
165000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G4A |
3-((1-benzhydryl-6-chloro-1H-indol-3-yl)methyl)-2-methoxybenzoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G4A |
4-(2-Hydroxy-3-{4-[(5-phenylpentyl)sulfanyl]phenoxy}propoxy)benzoic acid |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G4A |
4-((1-benzhydryl-6-chloro-1H-indol-3-yl)methyl)-3-methoxybenzoic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLA2G7 |
(2E)-2-[(7aS)-3-oxo-5,6,7,7a-tetrahydropyrrolo[1,2-c][1,3]oxazol-1-ylidene]acetic acid |
NA |
1700000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PLA2G7 |
(2,5-Dihydro-1h-Pyrrol-1-Yl)(3-Fluorophenyl)methanone |
NA |
NA|500000|5e+05 |
980000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PLA2G7 |
1,3-Dimethyl-6-(2-Methylpropoxy)pyrimidine-2,4(1h,3h)-Dione |
NA |
1000000|1e+06 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PLA2G7 |
1-Methyl-3-(2-phenoxyethyl)imidazolidine-2,4-dione |
NA |
1000000|1e+06 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PLA2G7 |
5,5-Dimethylhydantoin |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLA2G7 |
Methanesulfonamide, N-(3,4-difluorophenyl)- |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLA2G7 |
Abx-1431 |
NA |
494000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PLA2G7 |
Benzenesulfonamide |
NA |
NA|1000000 |
3400000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PLAT |
N-(3-Bromo-5-chloro-pyridin-2-yl)-guanidine |
272000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
|
165000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAT |
H-Cys(1)-Pro-Ala-Tyr-Ser-Arg-Tyr-Leu-Asp-Cys(1)-OH |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
(S)-1-(3,3-Diphenyl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
(2S)-N-cyclopentyl-N-methyl-5-[4-(methylamino)phenyl]-2-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonylamino)pent-4-ynamide |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |