| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAT |
1-(2-Amino-3,3-dicyclohexyl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide |
137000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
(2S)-N-cyclopentyl-N-methyl-5-[4-(methylamino)phenyl]-2-[(4-propylphenyl)sulfonylamino]pent-4-ynamide |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
Tfa-D-aMePhg-Pro-Arg-al |
NA |
30000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
4-[(2R)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]-N,N-dimethylpiperazine-1-carboxamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
Ac-D-aMePhg-Aze-Arg-al |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
3-[(R)-3-(4-Formyl-piperazin-1-yl)-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
3-[(R)-3-(4-Methyl-piperazin-1-yl)-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
(S)-1-(2-5H-Dibenzo[a,d]cyclohepten-5-yl-acetyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; hydrochloride |
268000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
3-[(R)-3-(4-Acetyl-piperazin-1-yl)-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
410000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
Tfa-D-aMePhg-Aze-Arg-al |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
{(R)-2-[2-((S)-1-Formyl-4-guanidino-butylcarbamoyl)-azetidin-1-yl]-1-methyl-2-oxo-1-phenyl-ethyl}-carbamic acid tert-butyl ester |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
3-[(R)-3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
3-[(R)-3-(4-Methanesulfonyl-piperazin-1-yl)-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
2-Biphenyl-3-yl-1H-indole-5-carboxamidine |
138000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
2-Phenyl-1H-benzoimidazole-5-carboxamidine |
381000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAT |
|
150000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAT |
2-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
[Benzyloxycarbonylamino-(4-guanidino-phenyl)-methyl]-phosphonic acid diphenyl ester trifluoro-acetic acid salt |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
(3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-amino-29-(4-aminobutyl)-11,23-dibenzyl-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-26-[3-(diaminomethylideneamino)propyl]-17-methyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
(3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-amino-11,23-dibenzyl-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-26-[3-(diaminomethylideneamino)propyl]-17,29-dimethyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |