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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAT Cycloleucine deriv. 43 108000 NA NA NA NA NA BindingDB|TTD
PLAT Diphenyl 1-(benzoylamino)-2-(4-guanidinophenyl)-ethanephosphonate NA 125000 NA NA NA NA BindingDB|TTD
PLAT N-Isoquinolin-1-yl-guanidine 126200 NA NA NA NA NA BindingDB|TTD
PLAT N-Quinolin-2-yl-guanidine 367000 NA NA NA NA NA BindingDB|TTD
PLAT Benzamidine 910000 NA NA NA NA NA BindingDB|TTD
PLAT 180000 NA NA NA NA NA BindingDB
PLAT [Amino({4-[(3-hydroxynaphthalene-2-)amido]phenyl}amino)methylidene]azanium 670000 NA NA NA NA NA BindingDB
PLAT 2-amino-5-[(2-hydroxy-3-phenylbenzene)amido]-1H-1,3-benzodiazol-3-ium 270000 NA NA NA NA NA BindingDB
PLAT N-(4-Carbamimidoyl-3-choro-phenyl)-2-hydroxy-3-iodo-5-methyl-benzamide 210000|256000 NA NA NA NA NA BindingDB|TTD
PLAT (2S)-N-cyclopentyl-N-methyl-5-[4-(methylamino)phenyl]-2-(naphthalen-2-ylsulfonylamino)pent-4-ynamide 200000 NA NA NA NA NA TTD
PLAT (2S)-N-cyclopentyl-2-[(6-methoxynaphthalen-2-yl)sulfonylamino]-N-methyl-5-[4-(methylamino)phenyl]pent-4-ynamide 200000 NA NA NA NA NA TTD
PLAT N-[5-Chloro-3-((E)-2-pyridin-2-yl-vinyl)-pyridin-2-yl]-guanidine 258500 NA NA NA NA NA BindingDB|TTD
PLAT N-(5-Chloro-3-phenoxy-pyridin-2-yl)-guanidine 342000 NA NA NA NA NA BindingDB|TTD
PLAT 225000 NA NA NA NA NA BindingDB
PLAT 263000 NA NA NA NA NA BindingDB
PLAT 150000 NA NA NA NA NA BindingDB
PLAT 425000 NA NA NA NA NA BindingDB
PLAT 275000 NA NA NA NA NA BindingDB
PLAT 3-Hydroxy-4-isopropoxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 563000 NA NA NA NA NA TTD
PLAT 3-Hydroxy-4-isopropoxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 300000 NA NA NA NA NA BindingDB|TTD