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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAT (S)-1-(3-Benzo[1,3]dioxol-5-yl-3-pyridin-3-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 500000 NA NA NA NA NA TTD
PLAT H-Tic-Pro-aMeArg-al NA 30000000 NA NA NA NA TTD
PLAT Me-Phe-Pro-aMeArg-al NA 30000000 NA NA NA NA TTD
PLAT tert-butyloxy carbonyl-D-Phe-DL-Pro(5,5-methyl)-Arg-H NA 30000000 NA NA NA NA TTD
PLAT N-[1-(3-Diaminomethyl-benzyl)-2-oxo-2-piperidin-1-yl-ethyl]-4-methyl-benzenesulfonamide 120000 NA NA NA NA NA BindingDB|TTD
PLAT (2S)-N-[(4-aminocyclohexyl)methyl]-1-[2-(benzylsulfonylamino)-3,3-diphenylpropanoyl]pyrrolidine-2-carboxamide 6700000 NA NA NA NA NA BindingDB|TTD
PLAT 2-(4-Guanidynephenyl)-1-phenyl-ethanone 1000000 NA NA NA NA NA TTD
PLAT (4-Guanidino-benzyl)-carbamic acid benzyl ester 1000000 NA NA NA NA NA TTD
PLAT [Amino(phenyl)methylidene]azanium 750000 NA NA NA NA NA BindingDB
PLAT 6-(N-Phenylcarbamyl)-2-Naphthalenecarboxamidine NA 125000 NA NA NA NA BindingDB
PLAT Thieno(2,3-B)Pyridine-2-Carboxamidine 1800000 NA NA NA NA NA BindingDB
PLAT Vaborbactam NA 1000000 NA NA NA NA PubChem|TTD
PLAT Benzyl 2-[(6-amino-5-carbamimidoyl-3-chloropyrazin-2-yl)amino]acetate NA 200000 NA NA NA NA BindingDB|TTD
PLAT Benzyl 2-[[6-amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetate NA 190000 NA NA NA NA TTD
PLAT 370000 NA NA NA NA NA BindingDB
PLAT 160000 NA NA NA NA NA BindingDB
PLAT 2-[(6-Amino-5-carbamimidoylpyrazin-2-yl)amino]acetic acid NA 250000 NA NA NA NA TTD
PLAT NA 200000 NA NA NA NA BindingDB
PLAT Benzyl 2-[(6-amino-5-carbamoyl-3-chloropyrazin-2-yl)amino]acetate NA 250000 NA NA NA NA TTD
PLAT 2-[(6-Amino-5-carbamimidoyl-3-chloropyrazin-2-yl)amino]acetic acid NA 250000 NA NA NA NA TTD