| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAT |
2-[[6-Amino-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[(2-aminoacetyl)amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]acetic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
(2S)-6-amino-2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[[(2S)-2-amino-3-hydroxypropanoyl]amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]hexanoic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAT |
3-[(2-Methylpropan-2-yl)oxycarbonylamino]propyl 3,4,5-trihydroxybenzoate |
NA |
581200 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAT |
2''-Sulfamoyl-biphenyl-4-carboxylic acid [2-(3-carbamimidoyl-phenoxy)-ethyl]-amide |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
2-Chloro-benzenesulfonic acid 3-methyl-5-[2-(methyl-pyridin-4-yl-amino)-ethoxy]-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetylamino]-3-(4-carbamimidoyl-phenyl)-propionic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
H-Cys(1)-Pro-Ala-Tyr-Ser-Arg-Tyr-Leu-Asp-Cys(1)-OH |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetylamino]-3-(4-carbamimidoyl-phenyl)-propionic acid ethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
3-(3-Carbamimidoyl-phenyl)-2-[2-(4-thiocarbamoyl-benzenesulfonylamino)-acetylamino]-propionic acid ethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
3-[(R)-3-(4-Methyl-piperazin-1-yl)-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
3-(4-Carbamimidoyl-phenyl)-2-[2-(4-cyano-benzenesulfonylamino)-acetylamino]-propionic acid ethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetylamino]-3-(3-carbamimidoyl-phenyl)-propionic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
3-(4-Carbamimidoyl-phenyl)-2-[2-(4-thiocarbamoyl-benzenesulfonylamino)-acetylamino]-propionic acid ethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
3-[(R)-3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
benzyl N-(4-amino-1-diphenoxyphosphorylbutyl)carbamate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
3-(3-Carbamimidoyl-phenyl)-2-[2-(4-cyano-benzenesulfonylamino)-acetylamino]-propionic acid ethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
5-[2-[3,4-Bis(hydroxymethyl)phenyl]-1,3-thiazol-4-yl]-1,3-dihydroindol-2-one |
NA |
205000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |