| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(4-pyridin-4-yloxyphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[[2,5-dioxo-3-(4-pyridin-4-yloxyphenyl)imidazolidin-1-yl]methyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-(2-Chloro-phenyl)-guanidine |
103000|103039 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
1-(Pyrimidin-2-yl)guanidine |
292000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
5-Amidinoindole |
131000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
3,5-Diamino-6-chloropyrazine-2-carbohydrazide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-(2-Methoxy-phenyl)-guanidine |
136000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-Pyrazinoylguanidine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[4-[[(2S)-2-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-3-phenylpropanoyl]amino]phenyl]acetic acid |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
(3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-amino-29-(4-aminobutyl)-11,23-dibenzyl-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-26-[3-(diaminomethylideneamino)propyl]-17-methyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
(3R,8S,11S,14S,17S,20S,23S,26S,29S,32S)-11-(4-acetamidobutyl)-3-amino-23-benzyl-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-26-[3-(diaminomethylideneamino)propyl]-17,29-dimethyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
methyl 2-[[4-[(2S)-2-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-3-(octylamino)-3-oxopropyl]phenoxy]methyl]benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
ethyl 4-[[4-[(2S)-2-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-3-(octylamino)-3-oxopropyl]phenoxy]methyl]benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
(3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-amino-11,23-dibenzyl-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-26-[3-(diaminomethylideneamino)propyl]-17,29-dimethyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
(3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-amino-23-benzyl-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-26-[3-(diaminomethylideneamino)propyl]-11-(1H-indol-3-ylmethyl)-17,29-dimethyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[4-[2-[(2-Ethylimidazo[1,2-a]pyridin-3-yl)amino]ethyl]phenyl]guanidine |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-[2-(2,4-dichlorophenoxy)ethyl]imidazo[1,2-a]pyridin-3-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-[4-(2-aminoethoxy)phenyl]imidazo[1,2-a]pyridin-3-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[4-(2-aminoethoxy)-3,5-dichlorophenyl]imidazo[1,2-a]pyridin-3-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
2-[4-[[(2-Pyridin-3-ylimidazo[1,2-a]pyridin-3-yl)amino]methyl]phenyl]guanidine |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |