Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAU H-D-Ser-Chg-Arg-OH (4) 321900 NA NA NA NA NA BindingDB
PLAU H-D-Ser-Cha-Arg-OH (5) 246970 NA NA NA NA NA BindingDB
PLAU H-D-Ser-homoCha-Arg-OH (6) 451200 NA NA NA NA NA BindingDB
PLAU H-D-Ser-alphaMePhe-Arg-OH (7) 275600 NA NA NA NA NA BindingDB
PLAU H-D-Ser-1ACH-Arg-OH (8) 395100 NA NA NA NA NA BindingDB
PLAU N-[2-[3,4-bis(hydroxymethyl)phenyl]ethyl]-2-hydrazinyl-2-oxoacetamide NA 2559000 NA NA NA NA BindingDB
PLAU 2-hydrazinyl-N-[[4-(hydroxymethyl)-2-methoxyphenyl]methyl]-2-oxoacetamide NA 2285000 NA NA NA NA BindingDB
PLAU 2-hydrazinyl-N-[[3-(hydroxymethyl)-5-methoxyphenyl]methyl]-2-oxoacetamide NA 4315000 NA NA NA NA BindingDB
PLAU 2-hydrazinyl-N-[(4-isocyanophenyl)methyl]-2-oxoacetamide NA 851000|892000|5469000 NA NA NA NA BindingDB
PLAU 2-Aminobenzimidazole NA 200000 NA NA NA NA BindingDB|TTD
PLAU 2-[[6-amino-5-[(Z)-N'-hydroxycarbamimidoyl]pyrazin-2-yl]amino]acetic acid NA 279000 NA NA NA NA TTD
PLAU 2-[[6-amino-3-chloro-5-[(Z)-N'-hydroxycarbamimidoyl]pyrazin-2-yl]amino]acetic acid NA 231000 NA NA NA NA TTD
PLAU Nicotinoylguanidine NA 1000000 NA NA NA NA TTD
PLAU Xeruborbactam NA 1000000 NA NA NA NA PubChem
PLAU Guanidinocarbonylpyridine NA 1000000 NA NA NA NA TTD
PLAU Methyl 4-guanidinobenzoate 1448771.85 NA NA NA NA NA TTD
PLAU (2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-fluorophenyl)sulfonylamino]acetamide NA 280000 NA NA NA NA BindingDB
PLAU (2R)-N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-2-phenylacetamide NA 140000 NA NA NA NA BindingDB|TTD
PLAU 5-H-Amiloride NA 1000000 NA NA NA NA TTD
PLAU 4-Guanidinobenzoic Acid 744732|745000|744731.97 NA NA NA NA NA BindingDB|TTD