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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAU 4-(4-Cyclohexyl-thiazol-2-yl)-5-methylsulfanyl-thiophene-2-carboxamidine 641000 NA NA NA NA NA TTD
PLAU 5-Methylsulfanyl-4-(4-naphthalen-2-yl-thiazol-2-yl)-thiophene-2-carboxamidine 138000 NA NA NA NA NA TTD
PLAU 5-Methylsulfanyl-4-(4-phenoxymethyl-thiazol-2-yl)-thiophene-2-carboxamidine 178000 NA NA NA NA NA TTD
PLAU 4-[4-(2,4-Dimethoxy-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 152000 NA NA NA NA NA TTD
PLAU 1-Methyl-1H-indole-5-carboximidamide 196000 NA NA NA NA NA BindingDB|TTD
PLAU 3-(3-Amino-1,2,4-oxadiazol-5-yl)-5-chloro-2,6-pyrazinediamine NA 1000000 NA NA NA NA TTD
PLAU N''-(2-Aminophenyl)guanidine 388000 NA NA NA NA NA TTD
PLAU N-Quinolin-2-yl-guanidine 209000 NA NA NA NA NA BindingDB|TTD
PLAU 3-(4-Guanidinophenyl)acrylic acid 1318256.74 NA NA NA NA NA TTD
PLAU Benzamidine 180000 NA NA NA NA NA BindingDB|TTD
PLAU 1-Ethyl-1H-indole-5-carboxamidine 280000 NA NA NA NA NA BindingDB|TTD
PLAU 1-Benzyl-1H-indole-5-carboxamidine 191000 NA NA NA NA NA BindingDB|TTD
PLAU Methyl 4-amino(immino)methylaminobenzoate 1448772|1450000 NA NA NA NA NA BindingDB
PLAU 2-(4-Methoxyphenyl)guanidine 676000|676083 NA NA NA NA NA BindingDB|TTD
PLAU 1N-amino(immino)methyl-2-methylaniline 258821|259000 NA NA NA NA NA BindingDB
PLAU 1N-amino(immino)methyl-2-methoxyaniline 136000|136144 NA NA NA NA NA BindingDB
PLAU N-o-tolyl-guanidine 258821.29 NA NA NA NA NA TTD
PLAU 2-Hydrazineyl-2-oxo-N-pentylacetamide NA 1933000 NA NA NA NA BindingDB
PLAU N-[(2-fluorophenyl)methyl]-2-hydrazinyl-2-oxoacetamide NA 1356000|1685000|2837000 NA NA NA NA BindingDB
PLAU N-(3-Fluorobenzyl)-2-hydrazinyl-2-oxoacetamide NA 1175000|1248000|2121000 NA NA NA NA BindingDB