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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAU (S)-ethyl 1-(5-(4-phenethoxybenzyl)-1,2,4-oxadiazol-3-yl)-6-amino-1-oxohexan-2-ylcarbamate 150000 NA NA NA NA NA TTD
PLAU Amiloride NA 107000 NA NA NA NA BindingDB|PubChem
PLAU 2-Amino-1H-benzimidazol-5-ol NA 200000 NA NA NA NA BindingDB|TTD
PLAU 2-hydrazinyl-N-[(4-methylphenyl)methyl]-2-oxoacetamide NA 229000|353000|533000 NA NA NA NA BindingDB
PLAU (2R)-1-(2,6-dimethylphenoxy)propan-2-amine NA 1000000 NA NA NA NA TTD
PLAU 5-Methylsulfanyl-4-(4-o-tolyl-thiazol-2-yl)-thiophene-2-carboxamidine 277000 NA NA NA NA NA TTD
PLAU 5-Methylsulfanyl-4-[4-(4-nitro-phenyl)-thiazol-2-yl]-thiophene-2-carboxamidine 270000 NA NA NA NA NA TTD
PLAU 4-[4-(4-Chloro-pyridin-3-yl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 164000 NA NA NA NA NA TTD
PLAU 5-Methylsulfanyl-4-(4-m-tolyl-thiazol-2-yl)-thiophene-2-carboxamidine 546000 NA NA NA NA NA TTD
PLAU 4-[4-(4-Methoxy-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 327000 NA NA NA NA NA TTD
PLAU 4-[4-(2-Chloro-pyridin-3-yl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 154000 NA NA NA NA NA TTD
PLAU 4-(4,5-Diphenyl-thiazol-2-yl)-5-methylsulfanyl-thiophene-2-carboxamidine 982000 NA NA NA NA NA TTD
PLAU 4-[4-(2-Chloro-pyridin-4-yl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 120000 NA NA NA NA NA TTD
PLAU 4-(4-Biphenyl-4-yl-thiazol-2-yl)-5-methylsulfanyl-thiophene-2-carboxamidine 1740000 NA NA NA NA NA TTD
PLAU 4-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 108000 NA NA NA NA NA TTD
PLAU 4-(4-Benzyl-thiazol-2-yl)-5-methylsulfanyl-thiophene-2-carboxamidine 470000 NA NA NA NA NA TTD
PLAU 4-[4-(2-Methoxy-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 130000 NA NA NA NA NA TTD
PLAU 4-[4-(3-Bromo-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 442000 NA NA NA NA NA TTD
PLAU 4-(5-Methyl-4-phenyl-thiazol-2-yl)-5-methylsulfanyl-thiophene-2-carboxamidine 305000 NA NA NA NA NA TTD
PLAU 4-[4-(4-Chloro-3-nitro-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine 161000 NA NA NA NA NA TTD