| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
2-[4-[[(2-Piperidin-4-ylimidazo[1,2-a]pyridin-3-yl)amino]methyl]phenyl]guanidine |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-[4-(aminomethyl)cyclohexyl]imidazo[1,2-a]pyridin-3-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
2-[4-[[[2-(4-Fluorophenyl)imidazo[1,2-a]pyridin-3-yl]amino]methyl]phenyl]guanidine |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
2-[4-(Imidazo[1,2-a]pyridin-3-ylamino)butyl]guanidine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
2-[4-[[[2-Pyridin-3-yl-6-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]amino]methyl]phenyl]guanidine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1R)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]ethyl]-3-methylbenzimidazole-5-carboxamide |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1S)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-2-methylpropyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1R)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-2-methylpropyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1R,2R)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-2-methylbutyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1S)-1-[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]ethyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1R)-1-[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]ethyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1S)-1-[2,5-dioxo-3-(4-pyridin-4-yloxyphenyl)imidazolidin-1-yl]ethyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1R)-1-[2,5-dioxo-3-(4-pyridin-4-yloxyphenyl)imidazolidin-1-yl]ethyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1S)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]ethyl]-3-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-2-[(1R)-1-[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]-3-methylbutyl]-3-methylbenzimidazole-5-carboxamide |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
H-D-Ser-Ala-Arg-NH-(CH2)7-NH2 (6) |
244000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
H-D-Ser-Ala-Arg-NH-(CH2)9-NH2 (8) |
293000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
H-D-Ser-Phg-Arg-OH (1) |
487800 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
H-D-Ser-Phe-Arg-OH (2) |
544000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
H-D-Ser-homoPhe-Arg-OH (3) |
565800 |
NA |
NA |
NA |
NA |
NA |
BindingDB |