| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
2-Hydrazinyl-2-oxo-N-(3-(trifluoromethyl)benzyl)acetamide |
NA |
111000|136000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
5-Methylsulfanyl-4-[4-(4-p-tolylsulfamoyl-phenyl)-thiazol-2-yl]-thiophene-2-carboxamidine |
272000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
5-Methylsulfanyl-4-[4-(5,6,7,8-tetrahydro-naphthalen-2-yl)-thiazol-2-yl]-thiophene-2-carboxamidine |
145000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
4-(4-Benzo[b]thiophen-3-yl-thiazol-2-yl)-5-methylsulfanyl-thiophene-2-carboxamidine |
141000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
[4-(4-Aminobutyl)-3,6,9-trioxo-2,5,8-triazabicyclo[8.3.1]tetradeca-1(14),10,12-trien-11-yl]methyl-methyl-phenylsulfanium |
500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-Chloro-benzenesulfonic acid 3-(5-guanidino-pentyloxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-Chloro-benzenesulfonic acid 3-(1-carbamimidoyl-piperidin-3-ylmethoxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-Chloro-benzenesulfonic acid 3-(3-guanidino-propoxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-Chloro-benzenesulfonic acid 3-(4-guanidino-butoxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-(3-Hydroxy-pyridin-2-yl)-guanidine |
147000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-(6-Methyl-pyridin-2-yl)-guanidine |
173000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
N-(5-Chloro-3-phenyl-pyridin-2-yl)-guanidine |
166300 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
3-Benzoyl-1H-indole-6-carboxamidine |
267000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
3-[4-amino(immino)methylaminophenyl]-(E)-2-propenoic acid |
1318257|1330000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
1N-amino(immino)methyl-1,2-benzenediamine |
388000|388150 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
4-(5-Nitro-indol-1-ylmethyl)-benzamidine |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
(2S)-1-[(2R)-2-amino-3,3-diphenylpropanoyl]-N-[1-(diaminomethylideneamino)-5,8-dioxo-8-piperidin-1-yloctan-4-yl]pyrrolidine-2-carboxamide |
494000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
3-(3-Diaminomethyl-phenyl)-N-methyl-2-[2-(naphthalene-2-sulfonylamino)-acetylamino]-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
naphth-2-ylsulfonyl-Gly-DL-Phe(CH(NH2)2)-piperidide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(2S)-6-amino-1-[5-[[4-[2-(3,4-dichlorophenyl)ethoxy]phenyl]methyl]-1,2,4-oxadiazol-3-yl]-1-oxohexan-2-yl]-3,4-difluorobenzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |