| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
2-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]ethanesulfonic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]ethylphosphonic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
3-[4-[(6-Cyanonaphthalene-2-carbonyl)amino]phenyl]benzoic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
3-amino-6-chloro-N-(diaminomethylidene)-5-(2H-tetrazol-5-ylmethylamino)pyrazine-2-carboxamide |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]methylphosphonic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-(diaminomethylidene)-1H-imidazole-5-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
5-amino-6-bromo-N-(diaminomethylidene)pyrazine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-(3,5-Dihydroxybenzoyl)oxyethyl 3,4-dihydroxybenzoate |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(4-bromophenyl)methyl]-2-hydrazinyl-2-oxoacetamide |
NA |
167000|294000|525000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
Ethyl 2-[(4-bromophenyl)methylamino]-2-oxoacetate |
NA |
526000|692500|3016500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
Ethyl 2-oxo-2-[[3-(trifluoromethyl)phenyl]methylamino]acetate |
NA |
3794000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-hydrazinyl-N-[(3-methoxyphenyl)methyl]-2-oxoacetamide |
NA |
736000|776000|1337000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
Ethyl 2-[(3-chlorophenyl)methylamino]-2-oxoacetate |
NA |
4018000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-(3-Chlorobenzyl)-2-hydrazinyl-2-oxoacetamide |
NA |
126000|219000|558500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-hydrazinyl-2-oxo-N-[[4-(trifluoromethyl)phenyl]methyl]acetamide |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
|
NA |
231000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-[(6-Amino-5-carbamimidoylpyrazin-2-yl)amino]acetic acid |
NA |
212000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
|
NA |
279000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-[(6-Amino-5-carbamimidoyl-3-chloropyrazin-2-yl)amino]acetic acid |
NA |
237000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLAU |
2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[(2-aminoacetyl)amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]acetic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |