| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
(2S)-6-amino-2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[[(2S)-2-amino-3-hydroxypropanoyl]amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]hexanoic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
Ethyl 2-((4-chloro-3-(trifluoromethyl)benzyl)amino)-2-oxoacetate |
NA |
214000|219500|1196500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
Methyl 4-[[4-fluoro-3-(trifluoromethyl)phenyl]methylamino]-4-oxobutanoate |
NA |
428000|476000|1438000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
Methyl 4-[[4-chloro-3-(trifluoromethyl)phenyl]methylamino]-4-oxobutanoate |
NA |
145000|161700|734800 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
Methyl 4-oxo-4-[[3-(trifluoromethyl)phenyl]methylamino]butanoate |
NA |
752000|1061000|2909000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-((4-Chloro-3-(trifluoromethyl)benzyl)amino)-2-oxoacetic acid |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-Hydrazineyl-2-oxo-N-(3-(trifluoromethoxy)benzyl)acetamide |
NA |
134500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-N'-hydroxyoxamide |
NA |
162500|168000|205000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(4-chloro-2-methylphenyl)methyl]-N'-hydroxyoxamide |
NA |
5491000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(3,5-difluorophenyl)methyl]-N'-(propan-2-ylideneamino)oxamide |
NA |
490000|532000|1196000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-4-hydrazinyl-4-oxobutanamide |
NA |
124000|142000|641000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-(4-chloro-3-(trifluoromethyl)benzyl)-N'-methoxyoxalamide |
NA |
329000|513000|693000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-N'-methoxy-N'-methyloxamide |
NA |
318000|345000|713000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-[2-(benzenesulfonyl)hydrazinyl]-N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-2-oxoacetamide |
NA |
189000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-2-hydrazinyl-2-oxoacetamide |
NA |
108000|116500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-2-hydrazinyl-2-oxoacetamide |
NA |
102500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(4-fluoro-3-methylphenyl)methyl]-2-hydrazinyl-2-oxoacetamide |
NA |
178500 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(4-chloro-2-methylphenyl)methyl]-2-hydrazinyl-2-oxoacetamide |
NA |
121000|158500|222000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-4-hydrazinyl-4-oxobutanamide |
NA |
304000|363000|1187000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
4-hydrazinyl-4-oxo-N-[[3-(trifluoromethyl)phenyl]methyl]butanamide |
NA |
733000|1099000|2725000 |
NA |
NA |
NA |
NA |
BindingDB |