| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
3,4-dihydroxy-N-[[3-(trifluoromethyl)phenyl]methyl]benzamide |
NA |
475000|533000|898000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
3-hydroxy-N-(4-hydroxyphenyl)sulfonyl-N-octylbenzenesulfonamide |
NA |
177250 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-(Aminoiminomethyl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
Imidazo[1,2-a]pyridin-3-amine,n-[4-(aminomethyl)phenyl]- |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-oxo-N-(2-phenylethyl)-1,3-dihydroindole-5-sulfonamide |
NA |
1288000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-2-oxo-3H-1,3,4-oxadiazole-5-carboxamide |
NA |
265000|306000|405000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
1-[[4-Chloro-3-(trifluoromethyl)phenyl]methyl]-3-hydroxyurea |
NA |
2481000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
5-[2-[2-[[2-Oxo-2-(2-oxo-1,3-dihydroindol-5-yl)ethyl]amino]ethylamino]acetyl]-1,3-dihydroindol-2-one |
NA |
163000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
|
NA |
181000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
(2S)-1-(3,4-dihydroxyphenyl)sulfonyl-N-phenylpyrrolidine-2-carboxamide |
NA |
552000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
2-hydrazinyl-2-oxo-N-[[4-(trifluoromethoxy)phenyl]methyl]acetamide |
NA |
256500|279000|1922000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-5-methyl-1,2-oxazole-4-carboxamide |
NA |
524500|566000|680000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-5-methyl-1,2-oxazole-3-carboxamide |
NA |
580000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
4-[(2-Tert-butyl-5-cyclopropyl-1,2,4-triazol-3-yl)methyl]benzene-1,2-diol |
NA |
1608000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
4-[(2-Tert-butyl-5-pentyl-1,2,4-triazol-3-yl)methyl]benzene-1,2-diol |
NA |
116460|124600 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(4-chloro-2-methylphenyl)methyl]-2-oxo-3H-1,3,4-oxadiazole-5-carboxamide |
NA |
238000|628000|739000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(3-fluoro-4-methylphenyl)methyl]-2-oxo-3H-1,3,4-oxadiazole-5-carboxamide |
NA |
403000|405000|1159000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[2-(3,4-dihydroxyphenyl)ethyl]benzenesulfonamide |
NA |
189600 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
5-[(3,4-Dihydroxyphenyl)sulfonylamino]pentanoic acid |
NA |
663000 |
NA |
NA |
NA |
NA |
BindingDB |