| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(3-carbamoyl-4-phenoxyphenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-[3-carbamoyl-4-(pyridin-4-ylmethoxy)phenyl]-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-fluorophenyl)-5-oxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-7-methyl-6-[[5-oxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]methyl]pyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-4-(4-phenoxyphenyl)piperazin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
4-[4-(3-Methoxy-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine |
115000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
5-Methylsulfanyl-4-(4-methyl-thiazol-2-yl)-thiophene-2-carboxamidine |
815000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
4-[4-(2,4-Dichloro-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine |
287000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
2-Chloro-benzenesulfonic acid 3-(1-carbamimidoyl-piperidin-4-ylmethoxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAUR |
cyclo[Arg-Cys(1)-Thr-Lys-Ser-Ile-Pro-Pro-Ile-Cys(1)-Phe-D-Pro-Asp-Gly] |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLAUR |
Oxaprozin |
NA |
NA |
113900 |
NA |
NA |
NA |
BindingDB |
| PLAUR |
8-Methyl-4-(4-morpholinylcarbonyl)-2-phenylquinoline |
NA |
141000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PLAUR |
3-[(3-Bromo-4-hydroxy-6-methyl-9,10-dioxoanthracen-1-yl)amino]benzoic acid |
NA |
146000 |
NA |
NA |
NA |
NA |
TTD |
| PLCB1 |
Alpha-methyl-4-carboxyphenylglycine, (+/-)- |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLCB1 |
(1R,2S,3S)-2-(Amino-carboxy-methyl)-3-phenyl-cyclopropanecarboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| PLCB3 |
2-(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)benzo[de]isoquinoline-1,3-dione |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
6-{[cyclohexyl(methyl)amino]methyl}-N-(2-ethoxyphenyl)-1,3,5-triazine-2,4-diamine |
NA |
122517 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
N-(4-benzamido-3-methylphenyl)-1,3-benzodioxole-5-carboxamide |
NA |
122480 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
N-(4-Benzoylamino-3-methyl-phenyl)-3-ethoxy-benzamide |
NA |
122382 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
N-[2-chloro-4-[(4-propan-2-yloxybenzoyl)amino]phenyl]furan-2-carboxamide |
NA |
122498 |
NA |
NA |
NA |
NA |
BindingDB |