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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLCB3 (2E)-3-{1-[3-(dipropylamino)-2-hydroxypropyl]-1H-indol-3-yl}-1-thien-2-ylprop-2-en-1-one NA 122460 NA NA NA NA BindingDB
PLCB3 3-(2-methoxyphenyl)-2-{[(tetrahydro-2-furanylmethyl)amino]methyl}-4(3H)-quinazolinone NA 122382 NA NA NA NA BindingDB
PLCB3 4-(5-(Furan-2-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)butanoic acid NA 122506 NA NA NA NA BindingDB
PLCB3 N-[1-(1-Cyclopentyl-1H-tetrazol-5-ylmethyl)-piperidin-4-yl]-2-methyl-benzamide NA 122493 NA NA NA NA BindingDB
PLCB3 N-(6-benzamido-4-methylpyridin-3-yl)thiophene-2-carboxamide NA 122469 NA NA NA NA BindingDB
PLCB3 N-(4-methoxyphenyl)-3-(2-thienyl)-6-(trifluoromethyl)thieno[3,2-b]pyridine-2-carboxamide NA 122457 NA NA NA NA BindingDB
PLCB3 5-(4-chlorophenyl)-1-phenyl-1H-pyrazol-4-yl phenyl sulfone NA 122478 NA NA NA NA BindingDB
PLCB3 5-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl phenyl sulfone NA 122506 NA NA NA NA BindingDB
PLCB3 4-methoxybenzyl 1H-1,2,4-triazol-3-yl sulfone NA 122506 NA NA NA NA BindingDB
PLCB3 N-(2,4-dichlorophenyl)-2-{[3-(trifluoromethyl)phenyl]sulfinyl}acetamide NA 122457 NA NA NA NA BindingDB
PLCB3 2H-1,4-Benzothiazin-3(4H)-one 1,1-dioxide NA 122579 NA NA NA NA BindingDB
PLCB3 N-[4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]phenyl]-2-(1,3-dioxoisoindol-2-yl)acetamide NA 122387 NA NA NA NA BindingDB
PLCB3 (5Z)-5-(furan-2-ylmethylidene)-3-pyridin-3-yl-2-sulfanylidene-1,3-thiazolidin-4-one NA 122443 NA NA NA NA BindingDB
PLCB3 3-[4-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoylamino]benzoic acid NA 122499 NA NA NA NA BindingDB
PLCB3 Sennoside A, analytical standard NA 108765 NA NA NA NA BindingDB
PLCB3 2,4-Dinitropyrimidinyl-2-thiophenol NA 122702 NA NA NA NA BindingDB
PLCB3 Methyl 2-[2-[(4-tert-butylbenzoyl)amino]propanoylamino]-3-(4-hydroxyphenyl)propanoate NA 122508 NA NA NA NA BindingDB
PLCB3 2-(2,5-diketospiro[imidazolidine-4,1''-tetralin]-1-yl)-N-homoveratryl-N-methyl-acetamide NA 122490 NA NA NA NA BindingDB
PLCB3 1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(E)-[(E)-3-(4-nitrophenyl)prop-2-enylidene]amino]thiourea NA 122506 NA NA NA NA BindingDB
PLCB3 (E)-4-(3-(5-(furan-2-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)propanamido)-2-hydroxybenzoic acid NA 122481 NA NA NA NA BindingDB